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Journal of Medicinal Chemistry|August 9, 2002
Synthesis and biological activities of cyclic lanthionine enkephalin analogues: delta-opioid receptor selective ligandsYosup Rew, Shelle Malkmus, Camilla Svensson, et al.
Journal of Medicinal Chemistry|July 5, 2013
Cyclic enkephalins with a diversely substituted guanidine bridge or a thiourea bridge: synthesis, biological and structural evaluationsYouness Touati-Jallabe, Engin Bojnik, Baptiste Legrand, et al.
Journal of Medicinal Chemistry|September 28, 2016
A Cyclic Tetrapeptide ("Cyclodal") and Its Mirror-Image Isomer Are Both High-Affinity μ Opioid Receptor AntagonistsGrazyna Weltrowska, Thi M-D Nguyen, Nga N Chung, et al.
ACS Medicinal Chemistry Letters|May 20, 2014
In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt<sup>1</sup>-DALDA AnaloguesSteven Ballet, Cecilia Betti, Alexandre Novoa, et al.
Journal of Medicinal Chemistry|March 19, 2011
Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonistSteven Ballet, Debby Feytens, Koen Buysse, et al.
ACS Medicinal Chemistry Letters|November 21, 2017
χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone ScaffoldsOlivier Van der Poorten, Robin Van Den Hauwe, Emilie Eiselt, et al.
Journal of Medicinal Chemistry|October 30, 2012
Variation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and BiodistributionAlexandre Novoa, Sylvia Van Dorpe, Evelien Wynendaele, et al.
Bioorganic & Medicinal Chemistry Letters|June 2, 2018
Chemical space screening around Phe<sup>3</sup> in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplingsTom Willemse, Emilie Eiselt, Karlijn Hollanders, et al.
ACS Chemical Neuroscience|July 13, 2017
Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury MiceJoanna Starnowska, Roberto Costante, Karel Guillemyn, et al.
Journal of Medicinal Chemistry|April 2, 2016
Bifunctional Peptide-Based Opioid Agonist-Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic PainKarel Guillemyn, Joanna Starnowska, Camille Lagard, et al.
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