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Proceedings of the National Academy of Sciences of the United States of America
|
July 11, 2012
Preparation of unnatural N-to-N and C-to-C protein fusions
Martin D Witte, Juan J Cragnolini, Stephanie K Dougan, et al.
Journal of the American Chemical Society
|
July 21, 2009
Site-specific N- and C-terminal labeling of a single polypeptide using sortases of different specificity
John M Antos, Guo-Liang Chew, Carla P Guimaraes, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 28, 2019
Design, synthesis and evaluation of novel, potent DNA alkylating agents and their antibody-drug conjugates (ADCs)
Emily E Reid, Katie E Archer, Manami Shizuka, et al.
Bioconjugate Chemistry
|
November 21, 2019
Site-Specific Conjugation of the Indolinobenzodiazepine DGN549 to Antibodies Affords Antibody-Drug Conjugates with an Improved Therapeutic Index as Compared with Lysine Conjugation
Chen Bai, Emily E Reid, Alan Wilhelm, et al.
Bioconjugate Chemistry
|
May 14, 2016
Understanding How the Stability of the Thiol-Maleimide Linkage Impacts the Pharmacokinetics of Lysine-Linked Antibody-Maytansinoid Conjugates
Jose F Ponte, Xiuxia Sun, Nicholas C Yoder, et al.
Mabs
|
January 12, 2016
Microscale screening of antibody libraries as maytansinoid antibody-drug conjugates
Kalli C Catcott, Molly A McShea, Carl Uli Bialucha, et al.
Molecular Pharmaceutics
|
July 10, 2019
A Case Study Comparing Heterogeneous Lysine- and Site-Specific Cysteine-Conjugated Maytansinoid Antibody-Drug Conjugates (ADCs) Illustrates the Benefits of Lysine Conjugation
Nicholas C Yoder, Chen Bai, Daniel Tavares, et al.
Blood Advances
|
April 18, 2018
A CD123-targeting antibody-drug conjugate, IMGN632, designed to eradicate AML while sparing normal bone marrow cells
Yelena Kovtun, Gregory E Jones, Sharlene Adams, et al.
ACS Medicinal Chemistry Letters
|
August 16, 2019
Effect of Linker Stereochemistry on the Activity of Indolinobenzodiazepine Containing Antibody-Drug Conjugates (ADCs)
Emily E Reid, Katie E Archer, Manami Shizuka, et al.
Bioconjugate Chemistry
|
April 9, 2017
Effects of Drug-Antibody Ratio on Pharmacokinetics, Biodistribution, Efficacy, and Tolerability of Antibody-Maytansinoid Conjugates
Xiuxia Sun, Jose F Ponte, Nicholas C Yoder, et al.
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Search research articles
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Showing results (11-20 of 23) with videos related to
Sort By:
Page
of 3
Proceedings of the National Academy of Sciences of the United States of America
|
July 11, 2012
Preparation of unnatural N-to-N and C-to-C protein fusions
Martin D Witte, Juan J Cragnolini, Stephanie K Dougan, et al.
Journal of the American Chemical Society
|
July 21, 2009
Site-specific N- and C-terminal labeling of a single polypeptide using sortases of different specificity
John M Antos, Guo-Liang Chew, Carla P Guimaraes, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 28, 2019
Design, synthesis and evaluation of novel, potent DNA alkylating agents and their antibody-drug conjugates (ADCs)
Emily E Reid, Katie E Archer, Manami Shizuka, et al.
Bioconjugate Chemistry
|
November 21, 2019
Site-Specific Conjugation of the Indolinobenzodiazepine DGN549 to Antibodies Affords Antibody-Drug Conjugates with an Improved Therapeutic Index as Compared with Lysine Conjugation
Chen Bai, Emily E Reid, Alan Wilhelm, et al.
Bioconjugate Chemistry
|
May 14, 2016
Understanding How the Stability of the Thiol-Maleimide Linkage Impacts the Pharmacokinetics of Lysine-Linked Antibody-Maytansinoid Conjugates
Jose F Ponte, Xiuxia Sun, Nicholas C Yoder, et al.
Mabs
|
January 12, 2016
Microscale screening of antibody libraries as maytansinoid antibody-drug conjugates
Kalli C Catcott, Molly A McShea, Carl Uli Bialucha, et al.
Molecular Pharmaceutics
|
July 10, 2019
A Case Study Comparing Heterogeneous Lysine- and Site-Specific Cysteine-Conjugated Maytansinoid Antibody-Drug Conjugates (ADCs) Illustrates the Benefits of Lysine Conjugation
Nicholas C Yoder, Chen Bai, Daniel Tavares, et al.
Blood Advances
|
April 18, 2018
A CD123-targeting antibody-drug conjugate, IMGN632, designed to eradicate AML while sparing normal bone marrow cells
Yelena Kovtun, Gregory E Jones, Sharlene Adams, et al.
ACS Medicinal Chemistry Letters
|
August 16, 2019
Effect of Linker Stereochemistry on the Activity of Indolinobenzodiazepine Containing Antibody-Drug Conjugates (ADCs)
Emily E Reid, Katie E Archer, Manami Shizuka, et al.
Bioconjugate Chemistry
|
April 9, 2017
Effects of Drug-Antibody Ratio on Pharmacokinetics, Biodistribution, Efficacy, and Tolerability of Antibody-Maytansinoid Conjugates
Xiuxia Sun, Jose F Ponte, Nicholas C Yoder, et al.
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