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Cell Stress & Chaperones|May 23, 2021
Iso-mukaadial acetate and ursolic acid acetate inhibit the chaperone activity of Plasmodium falciparum heat shock protein 70-1Nicolaas Salomane, Ofentse J Pooe, Mthokozisi B C SimelaneScientific Reports|November 27, 2025
The impact of Iso-mukaadial acetate on Plasmodium falciparum transcriptional gene regulationNicolaas Salomane, Thendo Mafuna, Farhahna Allie, et al.Chemmedchem|February 16, 2026
Small Molecule Kinase Inhibitors with In Vitro β-Hematin Formation and Plasmodium falciparum Protein Kinase G Inhibitory Activity Identified Using Machine LearningJessica L Thibaud, Nicolaas Salomane, Sarah Harries, et al.Journal of Medicinal Chemistry|May 16, 2025
Medicinal Chemistry Progression of Sapanisertib, the Anticancer and Dual Plasmodium Phosphatidylinositol 4-Kinase Beta and cGMP-Dependent Protein Kinase Inhibitor, for MalariaSamuel Gachuhi, Stephanie Kamunya, Stephen Fienberg, et al.Microbiology Resource Announcements|January 15, 2019
Draft Genome Sequences of Seven Chryseobacterium Type StrainsAndisiwe Matu, Adeline Lum Nde, Lize Oosthuizen, et al.Journal of Medicinal Chemistry|October 7, 2025
Optimization of 2,8-Diaryl-1,5-naphthyridines as Plasmodium falciparum Phosphatidylinositol 4-Kinase Inhibitors with Improved ADME Profiles and In Vivo EfficacyGodwin A Dziwornu, Donald Seanego, Stephen Fienberg, et al.Journal of Medicinal Chemistry|August 14, 2025
Novel Inhibitors of Plasmodium Phosphatidylinositol 4-kinase IIIβ with Low Propensity for Resistance: Life Cycle Stage Activity and In Vivo Efficacy in a Humanized Mouse Malaria Infection ModelGodwin A Dziwornu, Mmakwena M Mmonwa, Dina Coertzen, et al.Angewandte Chemie (International Ed. in English)|October 24, 2025
Targeting Aurora Kinases as Essential Cell-Cycle Regulators to Deliver Multi-Stage Antimalarials Against Plasmodium FalciparumHenrico Langeveld, Keletso Maepa, Marché Maree, et al.Journal of Medicinal Chemistry|June 25, 2024
2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of Plasmodium falciparum Phosphatidylinositol-4-kinase and Hemozoin Formation with In Vivo EfficacyGodwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, et al.Pageof 1