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Journal of Enzyme Inhibition and Medicinal Chemistry|October 27, 2018
Refining the structure-activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoformsJoana Magalhães, Nina Franko, Giannamaria Annunziato, et al.
Pharmaceuticals (Basel, Switzerland)|June 24, 2022
Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative BacteriaGiannamaria Annunziato, Costanza Spadini, Marialaura Marchetti, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|September 18, 2018
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug designJoana Magalhães, Nina Franko, Giannamaria Annunziato, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|September 1, 2016
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMRGiannamaria Annunziato, Marco Pieroni, Roberto Benoni, et al.
ACS Infectious Diseases|January 29, 2021
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin AdjuvantGiannamaria Annunziato, Costanza Spadini, Nina Franko, et al.
Frontiers in Toxicology|July 23, 2026
Preventing regrettable substitutions: a proposal for a tiered testing approach for BPA alternatives under the PARC initiativeKiara Aiello-Holden, Kristina Bartmann, Franca Maria Buratti, et al.
Frontiers in Toxicology|December 15, 2025
Hazard identification and characterization of leachable chemicals from plastic products - a new PARC projectHubert Dirven, Aleksandra Bogusz, Hans Bouwmeester, et al.
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