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ACS Medicinal Chemistry Letters|February 20, 2018
From RORγt Agonist to Two Types of RORγt Inverse AgonistsYonghui Wang, Wei Cai, Ting Tang, et al.Journal of Medicinal Chemistry|April 17, 2012
Discovery of novel 1,2,4-thiadiazole derivatives as potent, orally active agonists of sphingosine 1-phosphate receptor subtype 1 (S1P(1))Feng Ren, Guanghui Deng, Hailong Wang, et al.Journal of Medicinal Chemistry|March 5, 2004
Evaluation of potent and selective small-molecule antagonists for the CXCR2 chemokine receptorKatherine L Widdowson, John D Elliott, Daniel F Veber, et al.Bioorganic & Medicinal Chemistry|August 17, 2015
Discovery of N-(4-aryl-5-aryloxy-thiazol-2-yl)-amides as potent RORγt inverse agonistsYonghui Wang, Ting Yang, Qian Liu, et al.Drug Resistance Updates : Reviews and Commentaries in Antimicrobial and Anticancer Chemotherapy|March 29, 2023
A phosphoglycerate mutase 1 allosteric inhibitor overcomes drug resistance to EGFR-targeted therapy via disrupting IL-6/JAK2/STAT3 signaling pathway in lung adenocarcinomaQian Liang, Miaomiao Gong, Jing-Hua Zou, et al.Cancer Research|October 4, 2022
Metabolic and Nonmetabolic Functions of PSAT1 Coordinate Signaling Cascades to Confer EGFR Inhibitor Resistance and Drive Progression in Lung AdenocarcinomaMing-Yu Luo, Ye Zhou, Wei-Ming Gu, et al.ACS Medicinal Chemistry Letters|July 21, 2015
Discovery of Biaryl Amides as Potent, Orally Bioavailable, and CNS Penetrant RORγt InhibitorsYonghui Wang, Wei Cai, Yaobang Cheng, et al.ACS Medicinal Chemistry Letters|June 6, 2014
Discovery of Tertiary Amine and Indole Derivatives as Potent RORγt Inverse AgonistsTing Yang, Qian Liu, Yaobang Cheng, et al.The Journal of Pharmacology and Experimental Therapeutics|May 18, 2004
XP13512 [(+/-)-1-([(alpha-isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane acetic acid], a novel gabapentin prodrug: I. Design, synthesis, enzymatic conversion to gabapentin, and transport by intestinal solute transportersKenneth C Cundy, Russell Branch, Tania Chernov-Rogan, et al.Bioorganic & Medicinal Chemistry Letters|June 4, 2011
Pyridazine-derived γ-secretase modulatorsZehong Wan, Adrian Hall, Yun Jin, et al.Pageof 18