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Journal of the American Chemical Society|July 17, 2003
First asymmetric total synthesis of tetrodotoxinNorio Ohyabu, Toshio Nishikawa, Minoru IsobeBioorganic & Medicinal Chemistry|August 21, 2013
Design, synthesis, and structure-activity relationships of dihydrofuran-2-one and dihydropyrrol-2-one derivatives as novel benzoxazin-3-one-based mineralocorticoid receptor antagonistsTomoaki Hasui, Taiichi Ohra, Norio Ohyabu, et al.ACS Medicinal Chemistry Letters|March 17, 2022
Discovery of TAK-925 as a Potent, Selective, and Brain-Penetrant Orexin 2 Receptor AgonistTatsuhiko Fujimoto, Kentaro Rikimaru, Koichiro Fukuda, et al.Journal of Medicinal Chemistry|November 15, 2011
Identification of benzoxazin-3-one derivatives as novel, potent, and selective nonsteroidal mineralocorticoid receptor antagonistsTomoaki Hasui, Nobuyuki Matsunaga, Taiichi Ora, et al.Bioorganic & Medicinal Chemistry|September 5, 2014
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonistsTomoaki Hasui, Norio Ohyabu, Taiichi Ohra, et al.Journal of Medicinal Chemistry|October 21, 2025
Discovery of Pyrazole-Based Positron Emission Tomography Agent that Maps Histone Deacetylase 6 (HDAC6) in the Nonhuman Primate BrainTomoteru Yamasaki, Norio Ohyabu, Takeshi Wakabayashi, et al.Pageof 1