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Molecules (Basel, Switzerland)|July 24, 2021
Design, Synthesis and Antiparasitic Evaluation of Click PhospholipidsGeorge E Magoulas, Pantelis Afroudakis, Kalliopi Georgikopoulou, et al.ACS Medicinal Chemistry Letters|April 19, 2019
SAR Studies and Biological Characterization of a Chromen-4-one Derivative as an Anti-<i>Trypanosoma brucei</i> AgentChiara Borsari, Nuno Santarem, Sara Macedo, et al.Journal of Medicinal Chemistry|November 3, 2023
High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic AgentsPasquale Linciano, Antonio Quotadamo, Rosaria Luciani, et al.Parasites & Vectors|November 29, 2025
Insights on genomic profiles of drug resistance and virulence in a cohort of Leishmania infantum isolates from the Mediterranean areaMarina Carrasco-Martin, Joan Martí-Carreras, Marcel Gómez-Ponce, et al.Journal of Medicinal Chemistry|March 26, 2019
Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic InfectionsPasquale Linciano, Cecilia Pozzi, Lucia Dello Iacono, et al.Bioorganic Chemistry|May 27, 2023
Design, synthesis and biological evaluation of antiparasitic dinitroaniline-ether phospholipid hybridsMarina Roussaki, George E Magoulas, Theano Fotopoulou, et al.European Journal of Medicinal Chemistry|January 9, 2017
Methoxylated 2'-hydroxychalcones as antiparasitic hit compoundsChiara Borsari, Nuno Santarem, Juan Torrado, et al.European Journal of Medicinal Chemistry|September 23, 2019
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomicsChiara Borsari, María Dolores Jiménez-Antón, Julia Eick, et al.Journal of Medicinal Chemistry|July 15, 2016
Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic DrugsChiara Borsari, Rosaria Luciani, Cecilia Pozzi, et al.Elife|December 7, 2022
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growthLuca Costantino, Stefania Ferrari, Matteo Santucci, et al.Pageof 3