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Molecular Pharmacology
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October 25, 2011
Functional impact of allosteric agonist activity of selective positive allosteric modulators of metabotropic glutamate receptor subtype 5 in regulating central nervous system function
Meredith J Noetzel, Jerri M Rook, Paige N Vinson, et al.
ACS Chemical Neuroscience
|
August 8, 2018
Discovery of Tricyclic Triazolo- and Imidazopyridine Lactams as M<sub>1</sub> Positive Allosteric Modulators
Julie L Engers, Aaron M Bender, Jacob J Kalbfleisch, et al.
ACS Chemical Neuroscience
|
September 13, 2016
Prefrontal Cortex-Mediated Impairments in a Genetic Model of NMDA Receptor Hypofunction Are Reversed by the Novel M<sub>1</sub> PAM VU6004256
Michael D Grannan, Catharine A Mielnik, Sean P Moran, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 28, 2021
Discovery of structurally distinct tricyclic M<sub>4</sub> positive allosteric modulator (PAM) chemotypes - Part 2
Madeline F Long, Rory A Capstick, Paul K Spearing, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 18, 2012
Continued optimization of the MLPCN probe ML071 into highly potent agonists of the hM1 muscarinic acetylcholine receptor
Bruce J Melancon, Rocco D Gogliotti, James C Tarr, et al.
ACS Chemical Neuroscience
|
June 23, 2026
Discovery of VU6066098: A Selective and CNS-Penetrant mGlu<sub>2</sub> NAM with Robust Antidepressant-, Antipsychotic-, and Procognitive-like Activity in Rodents
Jeremy S Coleman, Rory A Capstick, Sichen Chang, et al.
ACS Chemical Neuroscience
|
November 23, 2012
Targeting selective activation of M(1) for the treatment of Alzheimer's disease: further chemical optimization and pharmacological characterization of the M(1) positive allosteric modulator ML169
James C Tarr, Mark L Turlington, Paul R Reid, et al.
ACS Chemical Neuroscience
|
September 24, 2024
Discovery of VU6016235: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M<sub>4</sub> Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)
Julie L Engers, Logan A Baker, Sichen Chang, et al.
ACS Chemical Neuroscience
|
April 28, 2018
A Novel M<sub>1</sub> PAM VU0486846 Exerts Efficacy in Cognition Models without Displaying Agonist Activity or Cholinergic Toxicity
Jerri M Rook, Jeanette L Bertron, Hyekyung P Cho, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2017
Challenges in the development of an M<sub>4</sub> PAM preclinical candidate: The discovery, SAR, and in vivo characterization of a series of 3-aminoazetidine-derived amides
James C Tarr, Michael R Wood, Meredith J Noetzel, et al.
Page
of 30
Search research articles
Search
Showing results (261-270 of 299) with videos related to
Sort By:
Page
of 30
Molecular Pharmacology
|
October 25, 2011
Functional impact of allosteric agonist activity of selective positive allosteric modulators of metabotropic glutamate receptor subtype 5 in regulating central nervous system function
Meredith J Noetzel, Jerri M Rook, Paige N Vinson, et al.
ACS Chemical Neuroscience
|
August 8, 2018
Discovery of Tricyclic Triazolo- and Imidazopyridine Lactams as M<sub>1</sub> Positive Allosteric Modulators
Julie L Engers, Aaron M Bender, Jacob J Kalbfleisch, et al.
ACS Chemical Neuroscience
|
September 13, 2016
Prefrontal Cortex-Mediated Impairments in a Genetic Model of NMDA Receptor Hypofunction Are Reversed by the Novel M<sub>1</sub> PAM VU6004256
Michael D Grannan, Catharine A Mielnik, Sean P Moran, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 28, 2021
Discovery of structurally distinct tricyclic M<sub>4</sub> positive allosteric modulator (PAM) chemotypes - Part 2
Madeline F Long, Rory A Capstick, Paul K Spearing, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 18, 2012
Continued optimization of the MLPCN probe ML071 into highly potent agonists of the hM1 muscarinic acetylcholine receptor
Bruce J Melancon, Rocco D Gogliotti, James C Tarr, et al.
ACS Chemical Neuroscience
|
June 23, 2026
Discovery of VU6066098: A Selective and CNS-Penetrant mGlu<sub>2</sub> NAM with Robust Antidepressant-, Antipsychotic-, and Procognitive-like Activity in Rodents
Jeremy S Coleman, Rory A Capstick, Sichen Chang, et al.
ACS Chemical Neuroscience
|
November 23, 2012
Targeting selective activation of M(1) for the treatment of Alzheimer's disease: further chemical optimization and pharmacological characterization of the M(1) positive allosteric modulator ML169
James C Tarr, Mark L Turlington, Paul R Reid, et al.
ACS Chemical Neuroscience
|
September 24, 2024
Discovery of VU6016235: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M<sub>4</sub> Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)
Julie L Engers, Logan A Baker, Sichen Chang, et al.
ACS Chemical Neuroscience
|
April 28, 2018
A Novel M<sub>1</sub> PAM VU0486846 Exerts Efficacy in Cognition Models without Displaying Agonist Activity or Cholinergic Toxicity
Jerri M Rook, Jeanette L Bertron, Hyekyung P Cho, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2017
Challenges in the development of an M<sub>4</sub> PAM preclinical candidate: The discovery, SAR, and in vivo characterization of a series of 3-aminoazetidine-derived amides
James C Tarr, Michael R Wood, Meredith J Noetzel, et al.
Page
of 30