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The Journal of Organic Chemistry|November 15, 2000
Enantiopure 4- and 5-aminopiperidin-2-ones: regiocontrolled synthesis and conformational characterization as bioactive beta-turn mimeticsK Weber, U Ohnmacht, P GmeinerOrganic Letters|May 18, 2000
Treatment of N,N-dibenzylamino alcohols with sulfonyl chloride leads to rearranged beta-chloro amines, precursors to beta-amino acids, and not to tetrahydroisoquinolinesK Weber, S Kuklinski, P GmeinerBioorganic & Medicinal Chemistry Letters|September 11, 2001
Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179)J Einsiedel, H Hübner, P GmeinerJournal of Medicinal Chemistry|November 23, 2000
Cyanoindole derivatives as highly selective dopamine D(4) receptor partial agonists: solid-phase synthesis, binding assays, and functional experimentsH Hübner, J Kraxner, P GmeinerJournal of Medicinal Chemistry|February 26, 2000
Conjugated enynes as nonaromatic catechol bioisosteres: synthesis, binding experiments, and computational studies of novel dopamine receptor agonists recognizing preferentially the D(3) subtypeH Hübner, C Haubmann, W Utz, et al.Archiv Der Pharmazie|October 1, 1992
Tricyclic azaergoline analogues: synthesis, structural modifications, and pharmacological studiesP Gmeiner, J Sommer, G Höfner, et al.Bioorganic & Medicinal Chemistry Letters|January 5, 1999
Beta-analogs of PLG (L-prolyl-L-leucyl-glycinamide): ex-chiral pool syntheses and dopamine D2 receptor modulating effectsC Thomas, U Ohnmacht, M Niger, et al.Journal of Medicinal Chemistry|August 10, 2001
Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213)S Löber, H Hübner, W Utz, et al.Bioorganic & Medicinal Chemistry Letters|September 15, 2000
Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: synthesis and dopamine receptor binding profilesJ Einsiedel, C Thomas, H Hübner, et al.Die Pharmazie|May 11, 1999
[3H]Pramipexole: a selective radioligand for the high affinity dopamine D2 receptor in bovine striatal membranesU Ohnmacht, C Tränkle, K Mohr, et al.Pageof 3