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Journal of Medicinal Chemistry|December 24, 2004
Design, synthesis, and pharmacological characterization of novel, potent NMDA receptor antagonistsPaola Conti, Marco De Amici, Giovanni Grazioso, et al.
British Journal of Cancer|February 12, 2019
Inhibition of SIRT1 deacetylase and p53 activation uncouples the anti-inflammatory and chemopreventive actions of NSAIDsGiulia Dell'Omo, Daniela Crescenti, Cristina Vantaggiato, et al.
Journal of Medicinal Chemistry|September 1, 2015
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic ActivityThomas C Eadsforth, Andrea Pinto, Rosaria Luciani, et al.
The Journal of Biological Chemistry|February 22, 2011
The glial glutamate transporter 1 (GLT1) is expressed by pancreatic beta-cells and prevents glutamate-induced beta-cell deathEliana S Di Cairano, Alberto M Davalli, Lucia Perego, et al.
European Journal of Medicinal Chemistry|September 5, 2025
From pan-active to parasite-selective antiparasitic agents: A scaffold hopping approachChiara Borsari, Nuno Santarem, Dina Coertzen, et al.
ACS Infectious Diseases|May 8, 2024
Discovery of 1,3,4-Oxadiazole Derivatives as Broad-Spectrum Antiparasitic AgentsAlexandra Ioana Corfu, Nuno Santarem, Sara Luelmo, et al.
Journal of Medicinal Chemistry|May 26, 2026
First-in-Class Covalent Inhibitors of PFKFB3: Discovery and Characterization in PDAC ModelsAlessandra Fiore, Antonio Scarano, Giulia Antonini, et al.
European Journal of Medicinal Chemistry|January 27, 2020
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaignPasquale Linciano, Gregorio Cullia, Chiara Borsari, et al.
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