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Journal of Medicinal Chemistry|March 23, 2016
Discovery of Entrectinib: A New 3-Aminoindazole As a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitorMaria Menichincheri, Elena Ardini, Paola Magnaghi, et al.Journal of Medicinal Chemistry|July 30, 2015
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer TherapyGianluca Papeo, Helena Posteri, Daniela Borghi, et al.Journal of Medicinal Chemistry|June 11, 2004
3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead findingPaolo Pevarello, Maria Gabriella Brasca, Raffaella Amici, et al.Journal of Medicinal Chemistry|January 1, 2009
First Cdc7 kinase inhibitors: pyrrolopyridinones as potent and orally active antitumor agents. 2. Lead discoveryMaria Menichincheri, Alberto Bargiotti, Jens Berthelsen, et al.Journal of Medicinal Chemistry|September 30, 2010
Cdc7 kinase inhibitors: 5-heteroaryl-3-carboxamido-2-aryl pyrroles as potential antitumor agents. 1. Lead findingMaria Menichincheri, Clara Albanese, Cristina Alli, et al.Pageof 4