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Expert Opinion on Therapeutic Patents|April 26, 2015
Quinazoline derivatives as anticancer drugs: a patent review (2011 - present)Séverine Ravez, Omar Castillo-Aguilera, Patrick Depreux, et al.The Prostate|September 25, 2004
Synergistic antiproliferative and apoptotic effects induced by mixed epidermal growth factor receptor inhibitor ZD1839 and nitric oxide donor in human prostatic cancer cell linesMurielle Mimeault, Nathalie Jouy, Patrick Depreux, et al.European Journal of Medicinal Chemistry|February 8, 2005
New antiproliferative benzoindolinothiazepines derivativesGuillaume Laconde, Patrick Depreux, Pascal Berthelot, et al.Biomolecules|January 10, 2017
DNA Methylation Targeting: The DNMT/HMT Crosstalk ChallengeOmar Castillo-Aguilera, Patrick Depreux, Ludovic Halby, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|March 13, 2010
Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancerAntonio Garofalo, Laurence Goossens, Amelie Lemoine, et al.Molecular Cancer Therapeutics|February 25, 2010
Cytotoxic effects induced by docetaxel, gefitinib, and cyclopamine on side population and nonside population cell fractions from human invasive prostate cancer cellsMurielle Mimeault, Sonny L Johansson, Jean-Pierre Henichart, et al.Bioorganic & Medicinal Chemistry Letters|March 1, 2011
Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitorsAntonio Garofalo, Laurence Goossens, Perrine Six, et al.European Journal of Medicinal Chemistry|April 22, 2014
Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitorsSéverine Ravez, Amélie Barczyk, Perrine Six, et al.Chirality|March 25, 2011
Preparative enantiomeric separation of new selective CB2 receptor agonists by liquid chromatography on polysaccharide-based chiral stationary phases: determination of enantiomeric purity and assignment of absolute stereochemistry by X-ray structure analysisEric Stern, Laurence Goossens, Pascal Retailleau, et al.Journal of Medicinal Chemistry|January 11, 2012
Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitorsAntonio Garofalo, Amaury Farce, Séverine Ravez, et al.Pageof 3