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Paul V Fish

Showing results (11-20 of 57) with videos related to

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Future Medicinal Chemistry|April 22, 2021
Small-molecule inhibitors of carboxylesterase NotumYuguang Zhao, Sarah Jolly, Stefano Benvegnu, et al.
Bioorganic & Medicinal Chemistry Letters|April 18, 2008
Pyridyl-phenyl ether monoamine reuptake inhibitors: Impact of lipophilicity on dual SNRI pharmacology and off-target promiscuityGavin A Whitlock, Paul V Fish, M Jonathan Fray, et al.
SLAS Discovery : Advancing Life Sciences R & D|August 19, 2020
Changing the HTS Paradigm: AI-Driven Iterative Screening for Hit FindingGabriel H S Dreiman, Magda Bictash, Paul V Fish, et al.
Bioorganic & Medicinal Chemistry Letters|February 3, 2007
N-Benzyl-N-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-amines as selective dual serotonin/noradrenaline reuptake inhibitorsPaul V Fish, M Jonathan Fray, Alan Stobie, et al.
Bioorganic & Medicinal Chemistry Letters|June 6, 2006
Structure-activity relationships of N-substituted piperazine amine reuptake inhibitorsM Jonathan Fray, Gerwyn Bish, Paul V Fish, et al.
Bioorganic & Medicinal Chemistry Letters|April 11, 2009
4-Piperidines and 3-pyrrolidines as dual serotonin and noradrenaline reuptake inhibitors: design, synthesis and structure-activity relationshipsPaul V Fish, Mark D Andrews, M Jonathan Fray, et al.
Bioorganic & Medicinal Chemistry Letters|July 16, 2008
N-Benzyl-N-(pyrrolidin-3-yl)carboxamides as a new class of selective dual serotonin/noradrenaline reuptake inhibitorsFlorian Wakenhut, Paul V Fish, M Jonathan Fray, et al.
Bioorganic & Medicinal Chemistry Letters|June 6, 2006
N-(1,2-diphenylethyl)piperazines: a new class of dual serotonin/noradrenaline reuptake inhibitorM Jonathan Fray, Gerwyn Bish, Alan D Brown, et al.
Beilstein Journal of Organic Chemistry|December 7, 2019
An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agentNicky J Willis, Elliott D Bayle, George Papageorgiou, et al.
Bioorganic & Medicinal Chemistry Letters|August 4, 2016
New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atomsSophie S Spurr, Elliott D Bayle, Wenyu Yu, et al.
Pageof 6

Showing results (11-20 of 57) with videos related to

Sort By:
Pageof 6
Future Medicinal Chemistry|April 22, 2021
Small-molecule inhibitors of carboxylesterase NotumYuguang Zhao, Sarah Jolly, Stefano Benvegnu, et al.
Bioorganic & Medicinal Chemistry Letters|April 18, 2008
Pyridyl-phenyl ether monoamine reuptake inhibitors: Impact of lipophilicity on dual SNRI pharmacology and off-target promiscuityGavin A Whitlock, Paul V Fish, M Jonathan Fray, et al.
SLAS Discovery : Advancing Life Sciences R & D|August 19, 2020
Changing the HTS Paradigm: AI-Driven Iterative Screening for Hit FindingGabriel H S Dreiman, Magda Bictash, Paul V Fish, et al.
Bioorganic & Medicinal Chemistry Letters|February 3, 2007
N-Benzyl-N-(tetrahydro-2H-pyran-4-yl)pyrrolidin-3-amines as selective dual serotonin/noradrenaline reuptake inhibitorsPaul V Fish, M Jonathan Fray, Alan Stobie, et al.
Bioorganic & Medicinal Chemistry Letters|June 6, 2006
Structure-activity relationships of N-substituted piperazine amine reuptake inhibitorsM Jonathan Fray, Gerwyn Bish, Paul V Fish, et al.
Bioorganic & Medicinal Chemistry Letters|April 11, 2009
4-Piperidines and 3-pyrrolidines as dual serotonin and noradrenaline reuptake inhibitors: design, synthesis and structure-activity relationshipsPaul V Fish, Mark D Andrews, M Jonathan Fray, et al.
Bioorganic & Medicinal Chemistry Letters|July 16, 2008
N-Benzyl-N-(pyrrolidin-3-yl)carboxamides as a new class of selective dual serotonin/noradrenaline reuptake inhibitorsFlorian Wakenhut, Paul V Fish, M Jonathan Fray, et al.
Bioorganic & Medicinal Chemistry Letters|June 6, 2006
N-(1,2-diphenylethyl)piperazines: a new class of dual serotonin/noradrenaline reuptake inhibitorM Jonathan Fray, Gerwyn Bish, Alan D Brown, et al.
Beilstein Journal of Organic Chemistry|December 7, 2019
An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agentNicky J Willis, Elliott D Bayle, George Papageorgiou, et al.
Bioorganic & Medicinal Chemistry Letters|August 4, 2016
New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atomsSophie S Spurr, Elliott D Bayle, Wenyu Yu, et al.
Pageof 6