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Molecules (Basel, Switzerland)|September 23, 2022
Design, Synthesis and Structure-Activity Relationships of Phenylalanine-Containing Peptidomimetics as Novel HIV-1 Capsid Binders Based on Ugi Four-Component ReactionXiangkai Ji, Jing Li, Prem Prakash Sharma, et al.Journal of Medical Virology|April 5, 2024
Discovery of low-molecular-weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stabilityXiangyi Jiang, Zhen Gao, Prem Prakash Sharma, et al.Science Immunology|November 15, 2024
Palmitoylation of TIM-3 promotes immune exhaustion and restrains antitumor immunityZhaoying Zhang, Caiyue Ren, Rong Xiao, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|November 13, 2023
A novel N-heterocycles substituted oseltamivir derivatives as potent inhibitors of influenza virus neuraminidase: discovery, synthesis and biological evaluationJiwei Zhang, Chuanfeng Liu, Ruifang Jia, et al.Journal of Medicinal Chemistry|May 6, 2026
Discovery of a Novel Thienopyrimidine Derivative as a Potent Dual URAT1/GLUT9 Inhibitor with Enhanced Urate-Lowering Efficacy, Superior Pharmacokinetics, and Favorable Safety Profile for Gout and HyperuricemiaQian Yang, Danhui Qi, Wenjie Ye, et al.Research Square|May 10, 2023
Targeting Sex Determination to Suppress Mosquito PopulationsOmar Akbari, Ming Li, Nikolay Kandul, et al.RSC Medicinal Chemistry|July 24, 2023
Design, synthesis, and mechanistic study of 2-piperazineone-bearing peptidomimetics as novel HIV capsid modulatorsXujie Zhang, Lin Sun, Shujing Xu, et al.Advanced Science (Weinheim, Baden-Wurttemberg, Germany)|September 15, 2025
Discovery of a Baloxavir-Inspired Endonuclease Inhibitor That Prevents Herpes Simplex Virus 1 Replication in Cell Culture and In VivoSabina Andreu, Kai Tang, Jiahui Zhou, et al.Bioorganic & Medicinal Chemistry|March 10, 2026
Novel antiviral compounds: Synthesis, biological studies on SARS-CoV-2, and structure-activity relationship analysisSumit Kumar, Renata Pessôa Germano Mendes, Meenakshi Bansal, et al.Journal of Medicinal Chemistry|November 22, 2023
Design, Synthesis, and Biological Evaluation of Trisubstituted Piperazine Derivatives as Noncovalent Severe Acute Respiratory Syndrome Coronavirus 2 Main Protease Inhibitors with Improved Antiviral Activity and Favorable DruggabilityShenghua Gao, Letian Song, Katharina Sylvester, et al.Pageof 56