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Journal of Medicinal Chemistry|May 27, 2005
Fancy bioisosteres: metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profilesKarin Schlotter, Frank Boeckler, Harald Hübner, et al.Journal of Medicinal Chemistry|June 9, 2006
Fancy bioisosteres: novel paracyclophane derivatives as super-affinity dopamine D3 receptor antagonistsKarin Schlotter, Frank Boeckler, Harald Hübner, et al.Bioorganic & Medicinal Chemistry|April 28, 2004
Clozapine derived 2,3-dihydro-1H-1,4- and 1,5-benzodiazepines with D4 receptor selectivity: synthesis and biological testingThomas Hussenether, Harald Hübner, Peter Gmeiner, et al.ACS Chemical Neuroscience|July 11, 2012
Engineering a GPCR-ligand pair that simulates the activation of D(2L) by DopamineNuska Tschammer, Miriam Dörfler, Harald Hübner, et al.Journal of Molecular Biology|November 1, 2011
Molecular dynamics simulations of the effect of the G-protein and diffusible ligands on the β2-adrenergic receptorAngela Goetz, Harald Lanig, Peter Gmeiner, et al.Bioorganic & Medicinal Chemistry|April 9, 2002
Phenylpiperazinylmethylindolecarboxylates and derivatives as selective D(4)-ligandsAnnette Moll, Harald Hübner, Peter Gmeiner, et al.Journal of Medicinal Chemistry|September 16, 2010
Bioisosteric replacement leading to biologically active [2.2]paracyclophanes with altered binding profiles for aminergic G-protein-coupled receptorsMarika Skultety, Harald Hübner, Stefan Löber, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|May 27, 2006
A highly practical RCM approach towards a molecular building kit of spirocyclic reverse turn mimicsHolger Bittermann, Frank Böckler, Jürgen Einsiedel, et al.Journal of Medicinal Chemistry|October 16, 2004
Evaluation of lactam-bridged neurotensin analogues adjusting psi(Pro10) close to the experimentally derived bioactive conformation of NT(8-13)Holger Bittermann, Jürgen Einsiedel, Harald Hübner, et al.Bioorganic & Medicinal Chemistry|July 2, 2017
Potent haloperidol derivatives covalently binding to the dopamine D2 receptorTobias Schwalbe, Jonas Kaindl, Harald Hübner, et al.Pageof 25