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Bioorganic & Medicinal Chemistry Letters|February 24, 2007
Synthesis and biological study of 2-amino-4-aryl-5-chloropyrimidine analogues as inhibitors of VEGFR-2 and cyclin dependent kinase 1 (CDK1)Shenlin Huang, Ronghua Li, Peter J Connolly, et al.Cancer Research|October 6, 2005
The in vitro and in vivo effects of JNJ-7706621: a dual inhibitor of cyclin-dependent kinases and aurora kinasesStuart Emanuel, Catherine A Rugg, Robert H Gruninger, et al.ACS Medicinal Chemistry Letters|August 23, 2021
Spirocyclic Thiohydantoin Antagonists of F877L and Wild-Type Androgen Receptor for Castration-Resistant Prostate CancerZhuming Zhang, Peter J Connolly, Luis Trabalón Escolar, et al.Bioorganic & Medicinal Chemistry Letters|August 6, 2008
A novel 5-[1,3,4-oxadiazol-2-yl]-N-aryl-4,6-pyrimidine diamine having dual EGFR/HER2 kinase activity: design, synthesis, and biological activityTerry V Hughes, Guozhang Xu, Steven K Wetter, et al.Journal of Medicinal Chemistry|July 8, 2005
Synthesis and identification of [1,3,5]triazine-pyridine biheteroaryl as a novel series of potent cyclin-dependent kinase inhibitorsGee-Hong Kuo, Alan Deangelis, Stuart Emanuel, et al.Bioorganic & Medicinal Chemistry Letters|January 4, 2015
A selective small molecule NOP (ORL-1 receptor) partial agonist for the treatment of anxietyTina Morgan Ross, Kathleen Battista, Gilles C Bignan, et al.Bioorganic & Medicinal Chemistry Letters|November 4, 2019
Discovery and optimization of a series of small-molecule allosteric inhibitors of MALT1 proteaseTianbao Lu, Peter J Connolly, Ulrike Philippar, et al.Biochemistry|January 27, 2010
Refolding and characterization of a soluble ectodomain complex of the calcitonin gene-related peptide receptorChristopher M Koth, Norzehan Abdul-Manan, Christopher A Lepre, et al.Journal of Medicinal Chemistry|March 18, 2005
Synthesis and discovery of pyrazine-pyridine biheteroaryl as a novel series of potent vascular endothelial growth factor receptor-2 inhibitorsGee-Hong Kuo, Aihua Wang, Stuart Emanuel, et al.Journal of Medicinal Chemistry|June 25, 2005
1-Acyl-1H-[1,2,4]triazole-3,5-diamine analogues as novel and potent anticancer cyclin-dependent kinase inhibitors: synthesis and evaluation of biological activitiesRonghui Lin, Peter J Connolly, Shenlin Huang, et al.Pageof 6