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Bioorganic & Medicinal Chemistry Letters|April 23, 2013
Novel adenosine A(2A) receptor ligands: a synthetic, functional and computational investigation of selected literature adenosine A(2A) receptor antagonists for extending into extracellular spaceManuela Jörg, Jeremy Shonberg, Frankie S Mak, et al.Journal of Medicinal Chemistry|October 22, 2013
A structure-activity analysis of biased agonism at the dopamine D2 receptorJeremy Shonberg, Carmen Klein Herenbrink, Laura López, et al.Journal of Medicinal Chemistry|June 12, 2018
Subtle Modifications to the Indole-2-carboxamide Motif of the Negative Allosteric Modulator N-(( trans)-4-(2-(7-Cyano-3,4-dihydroisoquinolin-2(1 H)-yl)ethyl)cyclohexyl)-1 H-indole-2-carboxamide (SB269652) Yield Dramatic Changes in Pharmacological Activity at the Dopamine D<sub>2</sub> ReceptorAnitha Kopinathan, Christopher Draper-Joyce, Monika Szabo, et al.ACS Chemical Neuroscience|February 19, 2016
Novel Fused Arylpyrimidinone Based Allosteric Modulators of the M1 Muscarinic Acetylcholine ReceptorShailesh N Mistry, Herman Lim, Manuela Jörg, et al.Chemical Communications (Cambridge, England)|January 8, 2014
Ionic liquids provide unique opportunities for oral drug delivery: structure optimization and in vivo evidence of utilityHywel D Williams, Yasemin Sahbaz, Leigh Ford, et al.Journal of Medicinal Chemistry|December 4, 2015
Synthesis, Biological Evaluation, and Utility of Fluorescent Ligands Targeting the μ-Opioid ReceptorLuke S Schembri, Leigh A Stoddart, Stephen J Briddon, et al.Journal of Medicinal Chemistry|April 29, 2009
Structure-guided design, synthesis, and evaluation of salicylic acid-based inhibitors targeting a selectivity pocket in the active site of human 20alpha-hydroxysteroid dehydrogenase (AKR1C1)Ossama El-Kabbani, Peter J Scammells, Joshua Gosling, et al.European Journal of Medicinal Chemistry|September 21, 2010
Structure-based optimization and biological evaluation of human 20α-hydroxysteroid dehydrogenase (AKR1C1) salicylic acid-based inhibitorsOssama El-Kabbani, Peter J Scammells, Tom Day, et al.Journal of Medicinal Chemistry|September 3, 2010
Effects of conformational restriction of 2-amino-3-benzoylthiophenes on A(1) adenosine receptor modulationLuigi Aurelio, Celine Valant, Bernard L Flynn, et al.British Journal of Pharmacology|October 10, 2019
The effect of two selective A<sub>1</sub> -receptor agonists and the bitopic ligand VCP746 on heart rate and regional vascular conductance in conscious ratsSamantha L Cooper, Julie March, Andrea R Sabbatini, et al.Pageof 15