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European Journal of Medicinal Chemistry
|
March 28, 2016
New IKK inhibitors: Synthesis of new imidazo[1,2-a]quinoxaline derivatives using microwave assistance and biological evaluation as IKK inhibitors
Georges Moarbess, Jean-François Guichou, Stéphanie Paniagua-Gayraud, et al.
Bioorganic & Medicinal Chemistry
|
February 26, 2004
Design and synthesis of novel imidazo[1,2-a]quinoxalines as PDE4 inhibitors
Carine Deleuze-Masquéfa, Grégori Gerebtzoff, Guy Subra, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences
|
October 27, 2009
Pharmacology of EAPB0203, a novel imidazo[1,2-a]quinoxaline derivative with anti-tumoral activity on melanoma
Sonia Khier, Carine Deleuze-Masquéfa, Georges Moarbess, et al.
European Journal of Medicinal Chemistry
|
December 14, 2020
Imidazo[1,2-a]quinoxalines for melanoma treatment with original mechanism of action
Cindy Patinote, Carine Deleuze-Masquéfa, Kamel Hadj Kaddour, et al.
Journal of Medicinal Chemistry
|
July 9, 2019
Novel and Selective TLR7 Antagonists among the Imidazo[1,2-<i>a</i>]pyrazines, Imidazo[1,5-<i>a</i>]quinoxalines, and Pyrazolo[1,5-<i>a</i>]quinoxalines Series
Nour Bou Karroum, Georges Moarbess, Jean-François Guichou, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
July 28, 2010
Metabolism and pharmacokinetics of EAPB0203 and EAPB0503, two imidazoquinoxaline compounds previously shown to have antitumoral activity on melanoma and T-lymphomas
Sonia Khier, Florence Gattacceca, Safia El Messaoudi, et al.
Biomedicines
|
June 27, 2024
Imiquimod Reverses Chronic Toxoplasmosis-Associated Behavioral and Neurocognitive Anomalies in a Rat Model
Shaymaa Itani, Maguy Hamie, Reem El Jammal, et al.
Biomolecules
|
May 28, 2025
The Novel Imiqualine EAPB02303 Is a Potent Drug for Treating Acute Myeloid Leukemia
Perla Makhoul, Rita Hleihel, Shaymaa Itani, et al.
Bioorganic & Medicinal Chemistry
|
April 21, 2016
New imidazoquinoxaline derivatives: Synthesis, biological evaluation on melanoma, effect on tubulin polymerization and structure-activity relationships
Zahraa Zghaib, Jean-François Guichou, Johanna Vappiani, et al.
Cell Death & Disease
|
June 9, 2025
Inhibiting microtubule polymerization with EAPB02303, a prodrug activated by catechol-O-methyl transferase, enhances paclitaxel effect in pancreatic cancer models
Kévin Bigot, Cindy Patinote, Véronique Garambois, et al.
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of 4
Search research articles
Search
Showing results (31-40 of 40) with videos related to
Sort By:
Page
of 4
You have reached the last page of results.
This site can display upto 40 results.
European Journal of Medicinal Chemistry
|
March 28, 2016
New IKK inhibitors: Synthesis of new imidazo[1,2-a]quinoxaline derivatives using microwave assistance and biological evaluation as IKK inhibitors
Georges Moarbess, Jean-François Guichou, Stéphanie Paniagua-Gayraud, et al.
Bioorganic & Medicinal Chemistry
|
February 26, 2004
Design and synthesis of novel imidazo[1,2-a]quinoxalines as PDE4 inhibitors
Carine Deleuze-Masquéfa, Grégori Gerebtzoff, Guy Subra, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences
|
October 27, 2009
Pharmacology of EAPB0203, a novel imidazo[1,2-a]quinoxaline derivative with anti-tumoral activity on melanoma
Sonia Khier, Carine Deleuze-Masquéfa, Georges Moarbess, et al.
European Journal of Medicinal Chemistry
|
December 14, 2020
Imidazo[1,2-a]quinoxalines for melanoma treatment with original mechanism of action
Cindy Patinote, Carine Deleuze-Masquéfa, Kamel Hadj Kaddour, et al.
Journal of Medicinal Chemistry
|
July 9, 2019
Novel and Selective TLR7 Antagonists among the Imidazo[1,2-<i>a</i>]pyrazines, Imidazo[1,5-<i>a</i>]quinoxalines, and Pyrazolo[1,5-<i>a</i>]quinoxalines Series
Nour Bou Karroum, Georges Moarbess, Jean-François Guichou, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
July 28, 2010
Metabolism and pharmacokinetics of EAPB0203 and EAPB0503, two imidazoquinoxaline compounds previously shown to have antitumoral activity on melanoma and T-lymphomas
Sonia Khier, Florence Gattacceca, Safia El Messaoudi, et al.
Biomedicines
|
June 27, 2024
Imiquimod Reverses Chronic Toxoplasmosis-Associated Behavioral and Neurocognitive Anomalies in a Rat Model
Shaymaa Itani, Maguy Hamie, Reem El Jammal, et al.
Biomolecules
|
May 28, 2025
The Novel Imiqualine EAPB02303 Is a Potent Drug for Treating Acute Myeloid Leukemia
Perla Makhoul, Rita Hleihel, Shaymaa Itani, et al.
Bioorganic & Medicinal Chemistry
|
April 21, 2016
New imidazoquinoxaline derivatives: Synthesis, biological evaluation on melanoma, effect on tubulin polymerization and structure-activity relationships
Zahraa Zghaib, Jean-François Guichou, Johanna Vappiani, et al.
Cell Death & Disease
|
June 9, 2025
Inhibiting microtubule polymerization with EAPB02303, a prodrug activated by catechol-O-methyl transferase, enhances paclitaxel effect in pancreatic cancer models
Kévin Bigot, Cindy Patinote, Véronique Garambois, et al.
Page
of 4