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Showing results (221-230 of 231) with videos related to

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Journal of Medicinal Chemistry|May 14, 2025
Diazepine Agonists of the 5-HT<sub>2C</sub> Receptor with Unprecedented Selectivity: Discovery of Bexicaserin (LP352)Albert Ren, Xiuwen Zhu, Juerg Lehmann, et al.
Bioorganic & Medicinal Chemistry Letters|April 6, 2010
Potent tricyclic pyrazole tetrazole agonists of the nicotinic acid receptor (GPR109a)P Douglas Boatman, Thomas O Schrader, Michelle Kasem, et al.
Bioorganic & Medicinal Chemistry Letters|January 24, 2012
Discovery of a second generation agonist of the orphan G-protein coupled receptor GPR119 with an improved profileGraeme Semple, Juerg Lehmann, Amy Wong, et al.
Journal of Medicinal Chemistry|June 12, 2023
Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC InteractionJian Ding, Lulu Liu, Ying-Ling Chiang, et al.
Bioorganic & Medicinal Chemistry Letters|March 30, 2011
Discovery of fused bicyclic agonists of the orphan G-protein coupled receptor GPR119 with in vivo activity in rodent models of glucose controlGraeme Semple, Albert Ren, Beatriz Fioravanti, et al.
Proceedings of the National Academy of Sciences of the United States of America|October 27, 1999
Attenuated sensitivity to neuroactive steroids in gamma-aminobutyrate type A receptor delta subunit knockout miceR M Mihalek, P K Banerjee, E R Korpi, et al.
ACS Chemical Biology|January 3, 2023
Discovery of Potent Small-Molecule Inhibitors of WDR5-MYC InteractionJian Ding, Guo Li, Hejun Liu, et al.
Journal of Medicinal Chemistry|July 31, 2008
3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): a partial agonist of the nicotinic acid receptor, G-protein coupled receptor 109a, with antilipolytic but no vasodilatory activity in miceGraeme Semple, Philip J Skinner, Tawfik Gharbaoui, et al.
Bioorganic & Medicinal Chemistry Letters|June 26, 2007
Agonist lead identification for the high affinity niacin receptor GPR109aTawfik Gharbaoui, Philip J Skinner, Young-Jun Shin, et al.
Journal of Medicinal Chemistry|March 23, 2012
(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (MK-1903): a potent GPR109a agonist that lowers free fatty acids in humansP Douglas Boatman, Brett Lauring, Thomas O Schrader, et al.
Pageof 24

Showing results (221-230 of 231) with videos related to

Sort By:
Pageof 24
Journal of Medicinal Chemistry|May 14, 2025
Diazepine Agonists of the 5-HT<sub>2C</sub> Receptor with Unprecedented Selectivity: Discovery of Bexicaserin (LP352)Albert Ren, Xiuwen Zhu, Juerg Lehmann, et al.
Bioorganic & Medicinal Chemistry Letters|April 6, 2010
Potent tricyclic pyrazole tetrazole agonists of the nicotinic acid receptor (GPR109a)P Douglas Boatman, Thomas O Schrader, Michelle Kasem, et al.
Bioorganic & Medicinal Chemistry Letters|January 24, 2012
Discovery of a second generation agonist of the orphan G-protein coupled receptor GPR119 with an improved profileGraeme Semple, Juerg Lehmann, Amy Wong, et al.
Journal of Medicinal Chemistry|June 12, 2023
Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC InteractionJian Ding, Lulu Liu, Ying-Ling Chiang, et al.
Bioorganic & Medicinal Chemistry Letters|March 30, 2011
Discovery of fused bicyclic agonists of the orphan G-protein coupled receptor GPR119 with in vivo activity in rodent models of glucose controlGraeme Semple, Albert Ren, Beatriz Fioravanti, et al.
Proceedings of the National Academy of Sciences of the United States of America|October 27, 1999
Attenuated sensitivity to neuroactive steroids in gamma-aminobutyrate type A receptor delta subunit knockout miceR M Mihalek, P K Banerjee, E R Korpi, et al.
ACS Chemical Biology|January 3, 2023
Discovery of Potent Small-Molecule Inhibitors of WDR5-MYC InteractionJian Ding, Guo Li, Hejun Liu, et al.
Journal of Medicinal Chemistry|July 31, 2008
3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): a partial agonist of the nicotinic acid receptor, G-protein coupled receptor 109a, with antilipolytic but no vasodilatory activity in miceGraeme Semple, Philip J Skinner, Tawfik Gharbaoui, et al.
Bioorganic & Medicinal Chemistry Letters|June 26, 2007
Agonist lead identification for the high affinity niacin receptor GPR109aTawfik Gharbaoui, Philip J Skinner, Young-Jun Shin, et al.
Journal of Medicinal Chemistry|March 23, 2012
(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (MK-1903): a potent GPR109a agonist that lowers free fatty acids in humansP Douglas Boatman, Brett Lauring, Thomas O Schrader, et al.
Pageof 24