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Journal of Medicinal Chemistry
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November 1, 2002
Discovery of gamma-lactam hydroxamic acids as selective inhibitors of tumor necrosis factor alpha converting enzyme: design, synthesis, and structure-activity relationships
James J-W Duan, Lihua Chen, Zelda R Wasserman, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 5, 2003
Nonbenzamidine tetrazole derivatives as factor Xa inhibitors
Mimi L Quan, Christopher D Ellis, Ming Y He, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 26, 2007
SAR and X-ray structures of enantiopure 1,2-cis-(1R,2S)-cyclopentyldiamine and cyclohexyldiamine derivatives as inhibitors of coagulation Factor Xa
Jennifer X Qiao, Chong-Hwan Chang, Daniel L Cheney, et al.
ACS Medicinal Chemistry Letters
|
November 19, 2021
Identification of 6-Hydroxypyrimidin-4(1<i>H</i>)-one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists
Zulan Pi, James A Johnson, Wei Meng, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 11, 2008
Sulfonamidolactam inhibitors of coagulation factor Xa
Joanne M Smallheer, Shuaige Wang, Mia L Laws, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 7, 2007
Structure-activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Donald J P Pinto, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 16, 2007
Design, structure-activity relationship, and pharmacokinetic profile of pyrazole-based indoline factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Irina C Jacobson, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 19, 2006
Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
Jennifer X Qiao, Xuhong Cheng, Joanne M Smallheer, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 27, 2001
Synthesis and SAR of benzamidine factor Xa inhibitors containing a vicinally-substituted heterocyclic core
J M Fevig, D J Pinto, Q Han, et al.
Bioorganic & Medicinal Chemistry
|
September 1, 1996
ACAT inhibitors derived from hetero-Diels-Alder cycloadducts of thioaldehydes
R G Wilde, J T Billheimer, S J Germain, et al.
Page
of 42
Search research articles
Search
Showing results (331-340 of 418) with videos related to
Sort By:
Page
of 42
Journal of Medicinal Chemistry
|
November 1, 2002
Discovery of gamma-lactam hydroxamic acids as selective inhibitors of tumor necrosis factor alpha converting enzyme: design, synthesis, and structure-activity relationships
James J-W Duan, Lihua Chen, Zelda R Wasserman, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 5, 2003
Nonbenzamidine tetrazole derivatives as factor Xa inhibitors
Mimi L Quan, Christopher D Ellis, Ming Y He, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 26, 2007
SAR and X-ray structures of enantiopure 1,2-cis-(1R,2S)-cyclopentyldiamine and cyclohexyldiamine derivatives as inhibitors of coagulation Factor Xa
Jennifer X Qiao, Chong-Hwan Chang, Daniel L Cheney, et al.
ACS Medicinal Chemistry Letters
|
November 19, 2021
Identification of 6-Hydroxypyrimidin-4(1<i>H</i>)-one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists
Zulan Pi, James A Johnson, Wei Meng, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 11, 2008
Sulfonamidolactam inhibitors of coagulation factor Xa
Joanne M Smallheer, Shuaige Wang, Mia L Laws, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 7, 2007
Structure-activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Donald J P Pinto, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 16, 2007
Design, structure-activity relationship, and pharmacokinetic profile of pyrazole-based indoline factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Irina C Jacobson, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 19, 2006
Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
Jennifer X Qiao, Xuhong Cheng, Joanne M Smallheer, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 27, 2001
Synthesis and SAR of benzamidine factor Xa inhibitors containing a vicinally-substituted heterocyclic core
J M Fevig, D J Pinto, Q Han, et al.
Bioorganic & Medicinal Chemistry
|
September 1, 1996
ACAT inhibitors derived from hetero-Diels-Alder cycloadducts of thioaldehydes
R G Wilde, J T Billheimer, S J Germain, et al.
Page
of 42