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Bioorganic & Medicinal Chemistry Letters
|
May 3, 2017
Neutral macrocyclic factor VIIa inhibitors
Nicholas R Wurtz, Brandon L Parkhurst, Indawati DeLucca, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2003
Rational design, synthesis and structure-activity relationships of a cyclic succinate series of TNF-alpha converting enzyme inhibitors. Part 2: lead optimization
Chu-Biao Xue, Xiaohua He, John Roderick, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 13, 2013
Nonbenzamidine acylsulfonamide tissue factor-factor VIIa inhibitors
Peter W Glunz, Xiaojun Zhang, Yan Zou, et al.
Journal of Medicinal Chemistry
|
January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide Linker
James R Corte, Tianan Fang, Honey Osuna, et al.
ACS Medicinal Chemistry Letters
|
June 16, 2022
Discovery of Heteroaryl Urea Isosteres for Formyl Peptide Receptor 2 Agonists
Nicholas R Wurtz, James A Johnson, Andrew Viet, et al.
Journal of Medicinal Chemistry
|
March 18, 2005
Discovery of 1-(3'-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2'-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide hydrochloride (razaxaban), a highly potent, selective, and orally bioavailable factor Xa inhibitor
Mimi L Quan, Patrick Y S Lam, Qi Han, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 15, 2020
Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa
Tianan Fang, James R Corte, Paul J Gilligan, et al.
Journal of Cardiovascular Pharmacology
|
August 13, 1998
Oral antiplatelet efficacy and specificity of a novel nonpeptide platelet GPIIb/IIIa receptor antagonist, DMP 802
S A Mousa, R E Olson, J M Bozarth, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 10, 2020
Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ
Michael C Myers, Donna M Bilder, Cullen L Cavallaro, et al.
Journal of Medicinal Chemistry
|
March 10, 2021
Discovery of a Hydroxypyridinone APJ Receptor Agonist as a Clinical Candidate
James A Johnson, Soong-Hoon Kim, Ji Jiang, et al.
Page
of 42
Search research articles
Search
Showing results (351-360 of 418) with videos related to
Sort By:
Page
of 42
Bioorganic & Medicinal Chemistry Letters
|
May 3, 2017
Neutral macrocyclic factor VIIa inhibitors
Nicholas R Wurtz, Brandon L Parkhurst, Indawati DeLucca, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2003
Rational design, synthesis and structure-activity relationships of a cyclic succinate series of TNF-alpha converting enzyme inhibitors. Part 2: lead optimization
Chu-Biao Xue, Xiaohua He, John Roderick, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 13, 2013
Nonbenzamidine acylsulfonamide tissue factor-factor VIIa inhibitors
Peter W Glunz, Xiaojun Zhang, Yan Zou, et al.
Journal of Medicinal Chemistry
|
January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide Linker
James R Corte, Tianan Fang, Honey Osuna, et al.
ACS Medicinal Chemistry Letters
|
June 16, 2022
Discovery of Heteroaryl Urea Isosteres for Formyl Peptide Receptor 2 Agonists
Nicholas R Wurtz, James A Johnson, Andrew Viet, et al.
Journal of Medicinal Chemistry
|
March 18, 2005
Discovery of 1-(3'-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2'-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide hydrochloride (razaxaban), a highly potent, selective, and orally bioavailable factor Xa inhibitor
Mimi L Quan, Patrick Y S Lam, Qi Han, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 15, 2020
Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa
Tianan Fang, James R Corte, Paul J Gilligan, et al.
Journal of Cardiovascular Pharmacology
|
August 13, 1998
Oral antiplatelet efficacy and specificity of a novel nonpeptide platelet GPIIb/IIIa receptor antagonist, DMP 802
S A Mousa, R E Olson, J M Bozarth, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 10, 2020
Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ
Michael C Myers, Donna M Bilder, Cullen L Cavallaro, et al.
Journal of Medicinal Chemistry
|
March 10, 2021
Discovery of a Hydroxypyridinone APJ Receptor Agonist as a Clinical Candidate
James A Johnson, Soong-Hoon Kim, Ji Jiang, et al.
Page
of 42