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Biochemical Pharmacology
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December 17, 2009
Reductive activation of the prodrug 1,2-bis(methylsulfonyl)-1-(2-chloroethyl)-2-[[1-(4-nitrophenyl)ethoxy]carbonyl]hydrazine (KS119) selectively occurs in oxygen-deficient cells and overcomes O(6)-alkylguanine-DNA alkyltransferase mediated KS119 tumor cell resistance
Raymond P Baumann, Philip G Penketh, Kimiko Ishiguro, et al.
Chemical Research in Toxicology
|
July 12, 2014
Influence of glutathione and glutathione S-transferases on DNA interstrand cross-link formation by 1,2-bis(methylsulfonyl)-1-(2-chloroethyl)hydrazine, the active anticancer moiety generated by laromustine
Philip G Penketh, Eric Patridge, Krishnamurthy Shyam, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 12, 2013
Chloroethylating and methylating dual function antineoplastic agents display superior cytotoxicity against repair proficient tumor cells
Rui Zhu, Raymond P Baumann, Eric Patridge, et al.
Chemical Biology & Drug Design
|
May 5, 2012
A strategy for selective O(6)-alkylguanine-DNA alkyltransferase depletion under hypoxic conditions
Philip G Penketh, Krishnamurthy Shyam, Raymond P Baumann, et al.
Analytical Biochemistry
|
May 19, 2016
When alcohol is the answer: Trapping, identifying and quantifying simple alkylating species in aqueous environments
Philip G Penketh, Krishnamurthy Shyam, Raymond P Baumann, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 31, 2012
Design of a hypoxia-activated prodrug inhibitor of O6-alkylguanine-DNA alkyltransferase
Rui Zhu, Helen A Seow, Raymond P Baumann, et al.
Journal of Cancer Therapy
|
August 16, 2013
Expression of <i>O</i><sup>6</sup>-Methylguanine-DNA Methyltransferase Examined by Alkyl-Transfer Assays, Methylation-Specific PCR and Western Blots in Tumors and Matched Normal Tissue
Kimiko Ishiguro, Krishnamurthy Shyam, Philip G Penketh, et al.
Journal of Medicinal Chemistry
|
September 30, 2011
4-nitrobenzyloxycarbonyl derivatives of O(6)-benzylguanine as hypoxia-activated prodrug inhibitors of O(6)-alkylguanine-DNA alkyltransferase (AGT), which produces resistance to agents targeting the O-6 position of DNA guanine
Rui Zhu, Mao-Chin Liu, Mei-Zhen Luo, et al.
Journal of Medicinal Chemistry
|
January 23, 2015
Antitumor sulfonylhydrazines: design, structure-activity relationships, resistance mechanisms, and strategies for improving therapeutic utility
Krishnamurthy Shyam, Philip G Penketh, Raymond P Baumann, et al.
Archives of Toxicology
|
June 7, 2012
7-Nitro-4-(phenylthio)benzofurazan is a potent generator of superoxide and hydrogen peroxide
Eric V Patridge, Emma S E Eriksson, Philip G Penketh, et al.
Page
of 3
Search research articles
Search
Showing results (11-20 of 24) with videos related to
Sort By:
Page
of 3
Biochemical Pharmacology
|
December 17, 2009
Reductive activation of the prodrug 1,2-bis(methylsulfonyl)-1-(2-chloroethyl)-2-[[1-(4-nitrophenyl)ethoxy]carbonyl]hydrazine (KS119) selectively occurs in oxygen-deficient cells and overcomes O(6)-alkylguanine-DNA alkyltransferase mediated KS119 tumor cell resistance
Raymond P Baumann, Philip G Penketh, Kimiko Ishiguro, et al.
Chemical Research in Toxicology
|
July 12, 2014
Influence of glutathione and glutathione S-transferases on DNA interstrand cross-link formation by 1,2-bis(methylsulfonyl)-1-(2-chloroethyl)hydrazine, the active anticancer moiety generated by laromustine
Philip G Penketh, Eric Patridge, Krishnamurthy Shyam, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 12, 2013
Chloroethylating and methylating dual function antineoplastic agents display superior cytotoxicity against repair proficient tumor cells
Rui Zhu, Raymond P Baumann, Eric Patridge, et al.
Chemical Biology & Drug Design
|
May 5, 2012
A strategy for selective O(6)-alkylguanine-DNA alkyltransferase depletion under hypoxic conditions
Philip G Penketh, Krishnamurthy Shyam, Raymond P Baumann, et al.
Analytical Biochemistry
|
May 19, 2016
When alcohol is the answer: Trapping, identifying and quantifying simple alkylating species in aqueous environments
Philip G Penketh, Krishnamurthy Shyam, Raymond P Baumann, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 31, 2012
Design of a hypoxia-activated prodrug inhibitor of O6-alkylguanine-DNA alkyltransferase
Rui Zhu, Helen A Seow, Raymond P Baumann, et al.
Journal of Cancer Therapy
|
August 16, 2013
Expression of <i>O</i><sup>6</sup>-Methylguanine-DNA Methyltransferase Examined by Alkyl-Transfer Assays, Methylation-Specific PCR and Western Blots in Tumors and Matched Normal Tissue
Kimiko Ishiguro, Krishnamurthy Shyam, Philip G Penketh, et al.
Journal of Medicinal Chemistry
|
September 30, 2011
4-nitrobenzyloxycarbonyl derivatives of O(6)-benzylguanine as hypoxia-activated prodrug inhibitors of O(6)-alkylguanine-DNA alkyltransferase (AGT), which produces resistance to agents targeting the O-6 position of DNA guanine
Rui Zhu, Mao-Chin Liu, Mei-Zhen Luo, et al.
Journal of Medicinal Chemistry
|
January 23, 2015
Antitumor sulfonylhydrazines: design, structure-activity relationships, resistance mechanisms, and strategies for improving therapeutic utility
Krishnamurthy Shyam, Philip G Penketh, Raymond P Baumann, et al.
Archives of Toxicology
|
June 7, 2012
7-Nitro-4-(phenylthio)benzofurazan is a potent generator of superoxide and hydrogen peroxide
Eric V Patridge, Emma S E Eriksson, Philip G Penketh, et al.
Page
of 3