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Rob Leurs

Showing results (91-100 of 285) with videos related to

Pageof 29
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Journal of Chemical Information and Modeling|June 17, 2008
Delineation of agonist binding to the human histamine H4 receptor using mutational analysis, homology modeling, and ab initio calculationsAldo Jongejan, Herman D Lim, Rogier A Smits, et al.
The Journal of Biological Chemistry|March 21, 2003
The carboxyl terminus of human cytomegalovirus-encoded 7 transmembrane receptor US28 camouflages agonism by mediating constitutive endocytosisMaria Waldhoer, Paola Casarosa, Mette M Rosenkilde, et al.
Journal of Medicinal Chemistry|July 21, 2006
Characterization of the histamine H4 receptor binding site. Part 1. Synthesis and pharmacological evaluation of dibenzodiazepine derivativesRogier A Smits, Herman D Lim, Bart Stegink, et al.
Journal of Medicinal Chemistry|August 15, 2013
KLIFS: a knowledge-based structural database to navigate kinase-ligand interaction spaceOscar P J van Linden, Albert J Kooistra, Rob Leurs, et al.
Journal of Medicinal Chemistry|February 25, 2016
PDEStrIAn: A Phosphodiesterase Structure and Ligand Interaction Annotated Database As a Tool for Structure-Based Drug DesignChimed Jansen, Albert J Kooistra, Georgi K Kanev, et al.
Molecular Pharmacology|November 17, 2023
Pharmacological Characterization of the Zebrafish (Danio Rerio) Histamine H<sub>1</sub> Receptor Reveals the Involvement of the Second Extracellular Loop in the Binding of HistamineDaniel A McNaught-Flores, Albert J Kooistra, Yu-Chia Chen, et al.
British Journal of Pharmacology|May 30, 2013
A single-point mutation (Ala280Val) in the third intracellular loop alters the signalling properties of the human histamine H₃ receptor stably expressed in CHO-K1 cellsCecilia Flores-Clemente, Angélica Osorio-Espinoza, Juan Escamilla-Sánchez, et al.
Biotechniques|November 25, 2010
An efficient and information-rich biochemical method design for fragment library screening on ion channelsAndrew J Thompson, Mark H P Verheij, Rob Leurs, et al.
Plos Neglected Tropical Diseases|September 16, 2017
The single cyclic nucleotide-specific phosphodiesterase of the intestinal parasite Giardia lamblia represents a potential drug targetStefan Kunz, Vreni Balmer, Geert Jan Sterk, et al.
European Journal of Pharmacology|December 9, 2003
Effects of clobenpropit on pentylenetetrazole-kindled seizures in ratsLisan Zhang, Zhong Chen, Keming Ren, et al.
Pageof 29

Showing results (91-100 of 285) with videos related to

Sort By:
Pageof 29
Journal of Chemical Information and Modeling|June 17, 2008
Delineation of agonist binding to the human histamine H4 receptor using mutational analysis, homology modeling, and ab initio calculationsAldo Jongejan, Herman D Lim, Rogier A Smits, et al.
The Journal of Biological Chemistry|March 21, 2003
The carboxyl terminus of human cytomegalovirus-encoded 7 transmembrane receptor US28 camouflages agonism by mediating constitutive endocytosisMaria Waldhoer, Paola Casarosa, Mette M Rosenkilde, et al.
Journal of Medicinal Chemistry|July 21, 2006
Characterization of the histamine H4 receptor binding site. Part 1. Synthesis and pharmacological evaluation of dibenzodiazepine derivativesRogier A Smits, Herman D Lim, Bart Stegink, et al.
Journal of Medicinal Chemistry|August 15, 2013
KLIFS: a knowledge-based structural database to navigate kinase-ligand interaction spaceOscar P J van Linden, Albert J Kooistra, Rob Leurs, et al.
Journal of Medicinal Chemistry|February 25, 2016
PDEStrIAn: A Phosphodiesterase Structure and Ligand Interaction Annotated Database As a Tool for Structure-Based Drug DesignChimed Jansen, Albert J Kooistra, Georgi K Kanev, et al.
Molecular Pharmacology|November 17, 2023
Pharmacological Characterization of the Zebrafish (Danio Rerio) Histamine H<sub>1</sub> Receptor Reveals the Involvement of the Second Extracellular Loop in the Binding of HistamineDaniel A McNaught-Flores, Albert J Kooistra, Yu-Chia Chen, et al.
British Journal of Pharmacology|May 30, 2013
A single-point mutation (Ala280Val) in the third intracellular loop alters the signalling properties of the human histamine H₃ receptor stably expressed in CHO-K1 cellsCecilia Flores-Clemente, Angélica Osorio-Espinoza, Juan Escamilla-Sánchez, et al.
Biotechniques|November 25, 2010
An efficient and information-rich biochemical method design for fragment library screening on ion channelsAndrew J Thompson, Mark H P Verheij, Rob Leurs, et al.
Plos Neglected Tropical Diseases|September 16, 2017
The single cyclic nucleotide-specific phosphodiesterase of the intestinal parasite Giardia lamblia represents a potential drug targetStefan Kunz, Vreni Balmer, Geert Jan Sterk, et al.
European Journal of Pharmacology|December 9, 2003
Effects of clobenpropit on pentylenetetrazole-kindled seizures in ratsLisan Zhang, Zhong Chen, Keming Ren, et al.
Pageof 29