Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Rob Leurs

Showing results (201-210 of 285) with videos related to

Pageof 29
Sort By:
Angewandte Chemie (International Ed. in English)|June 22, 2018
Photoswitching the Efficacy of a Small-Molecule Ligand for a Peptidergic GPCR: from Antagonism to AgonismXavier Gómez-Santacana, Sabrina M de Munnik, Prashanna Vijayachandran, et al.
The Journal of Biological Chemistry|October 3, 2003
Constitutive signaling of the human cytomegalovirus-encoded receptor UL33 differs from that of its rat cytomegalovirus homolog R33 by promiscuous activation of G proteins of the Gq, Gi, and Gs classesPaola Casarosa, Yvonne K Gruijthuijsen, Detlef Michel, et al.
Journal of Medicinal Chemistry|June 27, 2003
A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidineTakeshi Hashimoto, Shinya Harusawa, Lisa Araki, et al.
Journal of Medicinal Chemistry|October 19, 2011
Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studiesEnade P Istyastono, Saskia Nijmeijer, Herman D Lim, et al.
Journal of Biomolecular Screening|September 19, 2014
Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hitsAntoni R Blaazer, Kristina M Orrling, Anitha Shanmugham, et al.
Scientific Reports|January 27, 2018
Development of novel fluorescent histamine H<sub>1</sub>-receptor antagonists to study ligand-binding kinetics in living cellsLeigh A Stoddart, Andrea J Vernall, Monica Bouzo-Lorenzo, et al.
Journal of Immunology (Baltimore, Md. : 1950)|June 26, 2009
Significance of N-terminal proteolysis of CCL14a to activity on the chemokine receptors CCR1 and CCR5 and the human cytomegalovirus-encoded chemokine receptor US28Rudolf Richter, Paola Casarosa, Ludger Ständker, et al.
Molecular Pharmacology|September 25, 2019
Modulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, et al.
Beilstein Journal of Organic Chemistry|November 16, 2019
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with lightXavier Gómez-Santacana, Sabrina M de Munnik, Tamara A M Mocking, et al.
Proceedings of the National Academy of Sciences of the United States of America|July 15, 2024
Conformational dynamics underlying atypical chemokine receptor 3 activationOmolade Otun, Christelle Aljamous, Elise Del Nero, et al.
Pageof 29

Showing results (201-210 of 285) with videos related to

Sort By:
Pageof 29
Angewandte Chemie (International Ed. in English)|June 22, 2018
Photoswitching the Efficacy of a Small-Molecule Ligand for a Peptidergic GPCR: from Antagonism to AgonismXavier Gómez-Santacana, Sabrina M de Munnik, Prashanna Vijayachandran, et al.
The Journal of Biological Chemistry|October 3, 2003
Constitutive signaling of the human cytomegalovirus-encoded receptor UL33 differs from that of its rat cytomegalovirus homolog R33 by promiscuous activation of G proteins of the Gq, Gi, and Gs classesPaola Casarosa, Yvonne K Gruijthuijsen, Detlef Michel, et al.
Journal of Medicinal Chemistry|June 27, 2003
A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidineTakeshi Hashimoto, Shinya Harusawa, Lisa Araki, et al.
Journal of Medicinal Chemistry|October 19, 2011
Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studiesEnade P Istyastono, Saskia Nijmeijer, Herman D Lim, et al.
Journal of Biomolecular Screening|September 19, 2014
Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hitsAntoni R Blaazer, Kristina M Orrling, Anitha Shanmugham, et al.
Scientific Reports|January 27, 2018
Development of novel fluorescent histamine H<sub>1</sub>-receptor antagonists to study ligand-binding kinetics in living cellsLeigh A Stoddart, Andrea J Vernall, Monica Bouzo-Lorenzo, et al.
Journal of Immunology (Baltimore, Md. : 1950)|June 26, 2009
Significance of N-terminal proteolysis of CCL14a to activity on the chemokine receptors CCR1 and CCR5 and the human cytomegalovirus-encoded chemokine receptor US28Rudolf Richter, Paola Casarosa, Ludger Ständker, et al.
Molecular Pharmacology|September 25, 2019
Modulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, et al.
Beilstein Journal of Organic Chemistry|November 16, 2019
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with lightXavier Gómez-Santacana, Sabrina M de Munnik, Tamara A M Mocking, et al.
Proceedings of the National Academy of Sciences of the United States of America|July 15, 2024
Conformational dynamics underlying atypical chemokine receptor 3 activationOmolade Otun, Christelle Aljamous, Elise Del Nero, et al.
Pageof 29