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Rob Leurs

Showing results (231-240 of 285) with videos related to

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Journal of Medicinal Chemistry|July 6, 2019
Route to Prolonged Residence Time at the Histamine H<sub>1</sub> Receptor: Growing from Desloratadine to RupatadineReggie Bosma, Zhiyong Wang, Albert J Kooistra, et al.
Bioorganic & Medicinal Chemistry|March 4, 2016
Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidalsJohan Veerman, Toine van den Bergh, Kristina M Orrling, et al.
Journal of Medicinal Chemistry|November 16, 2012
Chemical subtleties in small-molecule modulation of peptide receptor function: the case of CXCR3 biaryl-type ligandsMaikel Wijtmans, Danny J Scholten, Luc Roumen, et al.
Journal of Medicinal Chemistry|September 11, 2010
Surface plasmon resonance biosensor based fragment screening using acetylcholine binding protein identifies ligand efficiency hot spots (LE hot spots) by deconstruction of nicotinic acetylcholine receptor α7 ligandsGerdien E de Kloe, Kim Retra, Matthis Geitmann, et al.
Antimicrobial Agents and Chemotherapy|December 28, 2020
Tetrahydrophthalazinone Inhibitor of Phosphodiesterase with <i>In Vitro</i> Activity against Intracellular TrypanosomatidsJulianna Siciliano de Araújo, Raiza Brandão Peres, Patrícia Bernardino da Silva, et al.
Journal of Medicinal Chemistry|May 15, 2013
Bispyrimidines as potent histamine H(4) receptor ligands: delineation of structure-activity relationships and detailed H(4) receptor binding modeHarald Engelhardt, Sabine Schultes, Chris de Graaf, et al.
Drug Discovery Today|December 26, 2012
Small and colorful stones make beautiful mosaics: fragment-based chemogenomicsChris de Graaf, Henry F Vischer, Gerdien E de Kloe, et al.
Molecular Pharmacology|September 28, 2011
Identification of a novel allosteric binding site in the CXCR2 chemokine receptorPetra de Kruijf, Herman D Lim, Luc Roumen, et al.
Cancer Research|March 26, 2009
The human cytomegalovirus-encoded chemokine receptor US28 promotes angiogenesis and tumor formation via cyclooxygenase-2David Maussang, Ellen Langemeijer, Carlos P Fitzsimons, et al.
European Journal of Medicinal Chemistry|March 20, 2012
Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonistsMaikel Wijtmans, David Maussang, Francesco Sirci, et al.
Pageof 29

Showing results (231-240 of 285) with videos related to

Sort By:
Pageof 29
Journal of Medicinal Chemistry|July 6, 2019
Route to Prolonged Residence Time at the Histamine H<sub>1</sub> Receptor: Growing from Desloratadine to RupatadineReggie Bosma, Zhiyong Wang, Albert J Kooistra, et al.
Bioorganic & Medicinal Chemistry|March 4, 2016
Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidalsJohan Veerman, Toine van den Bergh, Kristina M Orrling, et al.
Journal of Medicinal Chemistry|November 16, 2012
Chemical subtleties in small-molecule modulation of peptide receptor function: the case of CXCR3 biaryl-type ligandsMaikel Wijtmans, Danny J Scholten, Luc Roumen, et al.
Journal of Medicinal Chemistry|September 11, 2010
Surface plasmon resonance biosensor based fragment screening using acetylcholine binding protein identifies ligand efficiency hot spots (LE hot spots) by deconstruction of nicotinic acetylcholine receptor α7 ligandsGerdien E de Kloe, Kim Retra, Matthis Geitmann, et al.
Antimicrobial Agents and Chemotherapy|December 28, 2020
Tetrahydrophthalazinone Inhibitor of Phosphodiesterase with <i>In Vitro</i> Activity against Intracellular TrypanosomatidsJulianna Siciliano de Araújo, Raiza Brandão Peres, Patrícia Bernardino da Silva, et al.
Journal of Medicinal Chemistry|May 15, 2013
Bispyrimidines as potent histamine H(4) receptor ligands: delineation of structure-activity relationships and detailed H(4) receptor binding modeHarald Engelhardt, Sabine Schultes, Chris de Graaf, et al.
Drug Discovery Today|December 26, 2012
Small and colorful stones make beautiful mosaics: fragment-based chemogenomicsChris de Graaf, Henry F Vischer, Gerdien E de Kloe, et al.
Molecular Pharmacology|September 28, 2011
Identification of a novel allosteric binding site in the CXCR2 chemokine receptorPetra de Kruijf, Herman D Lim, Luc Roumen, et al.
Cancer Research|March 26, 2009
The human cytomegalovirus-encoded chemokine receptor US28 promotes angiogenesis and tumor formation via cyclooxygenase-2David Maussang, Ellen Langemeijer, Carlos P Fitzsimons, et al.
European Journal of Medicinal Chemistry|March 20, 2012
Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonistsMaikel Wijtmans, David Maussang, Francesco Sirci, et al.
Pageof 29