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Rob Leurs

Showing results (261-270 of 285) with videos related to

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Biochemical Pharmacology|April 3, 2025
Characterization of [<sup>3</sup>H]AZ12464237 as a high affinity, non-nucleotide antagonist radioligand for the P2Y<sub>12</sub> receptorE Johanna L Stéen, Efthalia-Natalia Tousiaki, Lee Kingston, et al.
Bioorganic & Medicinal Chemistry Letters|July 26, 2011
Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H₄ and the ion channel serotonin 5-HT₃AMark H P Verheij, Chris de Graaf, Gerdien E de Kloe, et al.
The Journal of Pharmacology and Experimental Therapeutics|February 5, 2009
Nonpeptidergic allosteric antagonists differentially bind to the CXCR2 chemokine receptorPetra de Kruijf, Jane van Heteren, Herman D Lim, et al.
Bioorganic & Medicinal Chemistry|May 6, 2009
Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studiesHerman D Lim, Enade P Istyastono, Andrea van de Stolpe, et al.
Journal of Medicinal Chemistry|April 25, 2008
4-benzyl-1H-imidazoles with oxazoline termini as histamine H3 receptor agonistsMaikel Wijtmans, Sylvain Celanire, Erwin Snip, et al.
Bioorganic & Medicinal Chemistry|August 6, 2019
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2)Erik de Heuvel, Abhimanyu K Singh, Pierre Boronat, et al.
Journal of the American Chemical Society|February 23, 2018
Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR PhotopharmacologyNiels J Hauwert, Tamara A M Mocking, Daniel Da Costa Pereira, et al.
Plos Neglected Tropical Diseases|July 31, 2020
Cloning and functional complementation of ten Schistosoma mansoni phosphodiesterases expressed in the mammalian host stagesJane C Munday, Stefan Kunz, Titilola D Kalejaiye, et al.
Chemmedchem|May 1, 2009
Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonistsSylvain Célanire, Maikel Wijtmans, Bernard Christophe, et al.
Antimicrobial Agents and Chemotherapy|July 1, 2020
Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruziJulianna Siciliano de Araújo, Cristiane França da Silva, Denise da Gama Jaén Batista, et al.
Pageof 29

Showing results (261-270 of 285) with videos related to

Sort By:
Pageof 29
Biochemical Pharmacology|April 3, 2025
Characterization of [<sup>3</sup>H]AZ12464237 as a high affinity, non-nucleotide antagonist radioligand for the P2Y<sub>12</sub> receptorE Johanna L Stéen, Efthalia-Natalia Tousiaki, Lee Kingston, et al.
Bioorganic & Medicinal Chemistry Letters|July 26, 2011
Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H₄ and the ion channel serotonin 5-HT₃AMark H P Verheij, Chris de Graaf, Gerdien E de Kloe, et al.
The Journal of Pharmacology and Experimental Therapeutics|February 5, 2009
Nonpeptidergic allosteric antagonists differentially bind to the CXCR2 chemokine receptorPetra de Kruijf, Jane van Heteren, Herman D Lim, et al.
Bioorganic & Medicinal Chemistry|May 6, 2009
Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studiesHerman D Lim, Enade P Istyastono, Andrea van de Stolpe, et al.
Journal of Medicinal Chemistry|April 25, 2008
4-benzyl-1H-imidazoles with oxazoline termini as histamine H3 receptor agonistsMaikel Wijtmans, Sylvain Celanire, Erwin Snip, et al.
Bioorganic & Medicinal Chemistry|August 6, 2019
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2)Erik de Heuvel, Abhimanyu K Singh, Pierre Boronat, et al.
Journal of the American Chemical Society|February 23, 2018
Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR PhotopharmacologyNiels J Hauwert, Tamara A M Mocking, Daniel Da Costa Pereira, et al.
Plos Neglected Tropical Diseases|July 31, 2020
Cloning and functional complementation of ten Schistosoma mansoni phosphodiesterases expressed in the mammalian host stagesJane C Munday, Stefan Kunz, Titilola D Kalejaiye, et al.
Chemmedchem|May 1, 2009
Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonistsSylvain Célanire, Maikel Wijtmans, Bernard Christophe, et al.
Antimicrobial Agents and Chemotherapy|July 1, 2020
Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruziJulianna Siciliano de Araújo, Cristiane França da Silva, Denise da Gama Jaén Batista, et al.
Pageof 29