Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Robert L Bertekap

Showing results (1-10 of 11) with videos related to

Pageof 2
Sort By:
Methods in Molecular Biology (Clifton, N.J.)|August 12, 2015
High-Throughput Screening for Allosteric Modulators of GPCRsRobert L Bertekap, Neil T Burford, Zhuyin Li, et al.
Assay and Drug Development Technologies|July 4, 2012
Development of a high-throughput calcium flux assay for identification of all ligand types including positive, negative, and silent allosteric modulators for G protein-coupled receptorsDevin J Noblin, Robert L Bertekap, Neil T Burford, et al.
Journal of Medicinal Chemistry|October 31, 2003
Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrileYong-Jin Wu, Huan He, Shuanghua Hu, et al.
Psychopharmacology|January 24, 2007
Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT 2A receptors: functional receptor-binding and in vivo electrophysiological studiesArlene D Stark, Shaun Jordan, Kelly A Allers, et al.
Bioorganic & Medicinal Chemistry|February 6, 2014
Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT₆ antagonistsShuanghua Hu, Yazhong Huang, Yong-Jin Wu, et al.
ACS Medicinal Chemistry Letters|December 21, 2016
Development of 1<i>H</i>-Pyrazolo[3,4-<i>b</i>]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric ModulatorsMatthew D Hill, Haiquan Fang, Jeffrey M Brown, et al.
Bioorganic & Medicinal Chemistry Letters|February 19, 2013
Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonistsIvar M McDonald, Robert A Mate, F Christopher Zusi, et al.
Bioorganic & Medicinal Chemistry Letters|September 4, 2007
Conformationally restricted homotryptamines. Part 4: Heterocyclic and naphthyl analogs of a potent selective serotonin reuptake inhibitorH Dalton King, Derek J Denhart, Jeffrey A Deskus, et al.
The Journal of Pharmacology and Experimental Therapeutics|November 20, 2015
Evidence for Classical Cholinergic Toxicity Associated with Selective Activation of M1 Muscarinic ReceptorsAndrew Alt, Annapurna Pendri, Robert L Bertekap, et al.
Bioorganic & Medicinal Chemistry Letters|December 21, 2012
Design, optimization, and in vivo evaluation of a series of pyridine derivatives with dual NK1 antagonism and SERT inhibition for the treatment of depressionKevin W Gillman, Michael F Parker, Mark Silva, et al.
Pageof 2

Showing results (1-10 of 11) with videos related to

Sort By:
Pageof 2
Methods in Molecular Biology (Clifton, N.J.)|August 12, 2015
High-Throughput Screening for Allosteric Modulators of GPCRsRobert L Bertekap, Neil T Burford, Zhuyin Li, et al.
Assay and Drug Development Technologies|July 4, 2012
Development of a high-throughput calcium flux assay for identification of all ligand types including positive, negative, and silent allosteric modulators for G protein-coupled receptorsDevin J Noblin, Robert L Bertekap, Neil T Burford, et al.
Journal of Medicinal Chemistry|October 31, 2003
Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrileYong-Jin Wu, Huan He, Shuanghua Hu, et al.
Psychopharmacology|January 24, 2007
Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT 2A receptors: functional receptor-binding and in vivo electrophysiological studiesArlene D Stark, Shaun Jordan, Kelly A Allers, et al.
Bioorganic & Medicinal Chemistry|February 6, 2014
Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT₆ antagonistsShuanghua Hu, Yazhong Huang, Yong-Jin Wu, et al.
ACS Medicinal Chemistry Letters|December 21, 2016
Development of 1<i>H</i>-Pyrazolo[3,4-<i>b</i>]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric ModulatorsMatthew D Hill, Haiquan Fang, Jeffrey M Brown, et al.
Bioorganic & Medicinal Chemistry Letters|February 19, 2013
Discovery of a novel series of quinolone α7 nicotinic acetylcholine receptor agonistsIvar M McDonald, Robert A Mate, F Christopher Zusi, et al.
Bioorganic & Medicinal Chemistry Letters|September 4, 2007
Conformationally restricted homotryptamines. Part 4: Heterocyclic and naphthyl analogs of a potent selective serotonin reuptake inhibitorH Dalton King, Derek J Denhart, Jeffrey A Deskus, et al.
The Journal of Pharmacology and Experimental Therapeutics|November 20, 2015
Evidence for Classical Cholinergic Toxicity Associated with Selective Activation of M1 Muscarinic ReceptorsAndrew Alt, Annapurna Pendri, Robert L Bertekap, et al.
Bioorganic & Medicinal Chemistry Letters|December 21, 2012
Design, optimization, and in vivo evaluation of a series of pyridine derivatives with dual NK1 antagonism and SERT inhibition for the treatment of depressionKevin W Gillman, Michael F Parker, Mark Silva, et al.
Pageof 2