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The Journal of Pharmacology and Experimental Therapeutics|February 20, 2014
Clinical and preclinical characterization of the histamine H(4) receptor antagonist JNJ-39758979Robin L Thurmond, Bin Chen, Paul J Dunford, et al.Inflammation Research : Official Journal of the European Histamine Research Society ... [Et Al.]|February 11, 2019
Toreforant, an orally active histamine H<sub>4</sub>-receptor antagonist, in patients with active rheumatoid arthritis despite methotrexate: mechanism of action results from a phase 2, multicenter, randomized, double-blind, placebo-controlled synovial biopsy studyDavid L Boyle, Samuel E DePrimo, Cesar Calderon, et al.The Journal of Experimental Medicine|August 3, 2005
Organic cation transporter 3 modulates murine basophil functions by controlling intracellular histamine levelsElke Schneider, François Machavoine, Jean-Marie Pléau, et al.The Journal of Pharmacology and Experimental Therapeutics|May 13, 2014
The histamine H₄ receptor antagonist, JNJ 39758979, is effective in reducing histamine-induced pruritus in a randomized clinical study in healthy subjectsAlexa Kollmeier, Klaus Francke, Bin Chen, et al.Bioorganic & Medicinal Chemistry Letters|January 18, 2015
Diaminopyrimidines, diaminopyridines and diaminopyridazines as histamine H4 receptor modulatorsBrad M Savall, Steven P Meduna, Kevin Tays, et al.Pharmacological Reviews|June 19, 2015
International Union of Basic and Clinical Pharmacology. XCVIII. Histamine ReceptorsPertti Panula, Paul L Chazot, Marlon Cowart, et al.The Journal of Pharmacology and Experimental Therapeutics|April 4, 2014
Histamine H4-receptors inhibit mast cell renin release in ischemia/reperfusion via protein kinase C ε-dependent aldehyde dehydrogenase type-2 activationSilvia Aldi, Ken-ichi Takano, Kengo Tomita, et al.Bioorganic & Medicinal Chemistry Letters|September 8, 2007
Pyrazole-based cathepsin S inhibitors with improved cellular potencyJianmei Wei, Barbara A Pio, Hui Cai, et al.Journal of Medicinal Chemistry|September 17, 2004
Nonpeptidic, noncovalent inhibitors of the cysteine protease cathepsin SRobin L Thurmond, Mary Pat Beavers, Hui Cai, et al.Bioorganic & Medicinal Chemistry Letters|December 3, 2014
The effect of pK(a) on pyrimidine/pyridine-derived histamine H4 ligandsBrad M Savall, Steven P Meduna, Jennifer Venable, et al.Pageof 8