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ACS Chemical Biology|July 7, 2012
Identification of small-molecule antagonists of the Pseudomonas aeruginosa transcriptional regulator PqsR: biophysically guided hit discovery and optimizationTobias Klein, Claudia Henn, Johannes C de Jong, et al.Journal of Medicinal Chemistry|March 18, 2005
Synthesis and evaluation of imidazolylmethylenetetrahydronaphthalenes and imidazolylmethyleneindanes: potent inhibitors of aldosterone synthaseSarah Ulmschneider, Ursula Müller-Vieira, Markus Mitrenga, et al.Journal of Medicinal Chemistry|July 10, 2013
Structure optimization of 2-benzamidobenzoic acids as PqsD inhibitors for Pseudomonas aeruginosa infections and elucidation of binding mode by SPR, STD NMR, and molecular dockingElisabeth Weidel, Johannes C de Jong, Christian Brengel, et al.Archiv Der Pharmazie|April 16, 2018
Design and synthesis of novel annulated thienopyrimidines as phosphodiesterase 5 (PDE5) inhibitorsLina Y El-Sharkawy, Rowaida A El-Sakhawy, Mohammad Abdel-Halim, et al.Journal of Medicinal Chemistry|February 26, 2015
Novel pyridyl substituted 4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolines as potent and selective aldosterone synthase inhibitors with improved in vitro metabolic stabilityQingzhong Hu, Lina Yin, Amjad Ali, et al.Journal of Medicinal Chemistry|October 16, 2008
Design, synthesis, biological evaluation and pharmacokinetics of bis(hydroxyphenyl) substituted azoles, thiophenes, benzenes, and aza-benzenes as potent and selective nonsteroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1)Emmanuel Bey, Sandrine Marchais-Oberwinkler, Ruth Werth, et al.Archiv Der Pharmazie|June 10, 2004
[1, 2-Bis(2, 6-difluoro-3-hydroxyphenyl)ethylene-diamine]platinum(II) complexes, compounds for the endocrine therapy of breast cancer - mode of action I: antitumor activity due to the reduction of the endogenous estrogen levelSabine Schertl, Rolf W Hartmann, Christine Batzl-Hartmann, et al.Journal of Medicinal Chemistry|July 18, 2008
Substituted 6-phenyl-2-naphthols. Potent and selective nonsteroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1): design, synthesis, biological evaluation, and pharmacokineticsSandrine Marchais-Oberwinkler, Patricia Kruchten, Martin Frotscher, et al.Journal of the American Chemical Society|August 19, 2017
Discovery of a Potent Inhibitor Class with High Selectivity toward Clostridial CollagenasesEsther Schönauer, Andreas M Kany, Jörg Haupenthal, et al.Journal of Cancer Research and Clinical Oncology|October 7, 2006
Platinum(II) complexes interfering with testicular steroid biosynthesis: drugs for the therapy of advanced or recurrent prostate cancers? Preclinical studiesSabine Schertl, Rolf W Hartmann, Christine Batzl-Hartmann, et al.Pageof 26