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Bioorganic & Medicinal Chemistry|July 15, 2009
Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profileRomano Silvestri, Alessia Ligresti, Giuseppe La Regina, et al.Archiv Der Pharmazie|November 22, 2023
Quinoline-based thiazolyl-hydrazones target cancer cells through autophagy inhibitionVladimir Ćurčić, Mateusz Olszewski, Natalia Maciejewska, et al.BMC Cancer|November 13, 2007
PYRROLO[1,2-b][1,2,5]BENZOTHIADIAZEPINES (PBTDs) induce apoptosis in K562 cellsGabriella Marfe, Carla Di Stefano, Romano Silvestri, et al.ACS Medicinal Chemistry Letters|October 16, 2020
Discovery of Zika Virus NS2B/NS3 Inhibitors That Prevent Mice from Life-Threatening Infection and Brain DamageAntonio Coluccia, Michela Puxeddu, Marianna Nalli, et al.Nature Chemical Biology|March 10, 2015
Pharmacological folding chaperones act as allosteric ligands of Frizzled4Serena F Generoso, Mariateresa Giustiniano, Giuseppe La Regina, et al.Neuro-Oncology|November 12, 2019
HDAC inhibition induces expression of scaffolding proteins critical for tumor progression in pediatric glioma: focus on EBP50 and IRSp53Caroline Capdevielle, Angélique Desplat, Justine Charpentier, et al.Journal of Medicinal Chemistry|February 11, 2015
Structure-based lead optimization and biological evaluation of BAX direct activators as novel potential anticancer agentsMariano Stornaiuolo, Giuseppe La Regina, Sara Passacantilli, et al.Bioorganic & Medicinal Chemistry Letters|January 7, 2023
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma bruceiKarol R Francisco, Ludovica Monti, Wenqian Yang, et al.Journal of Medicinal Chemistry|May 15, 2007
Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studiesGiuseppe La Regina, Michael C Edler, Andrea Brancale, et al.Cancers|March 10, 2022
Anticancer Activity of (S)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-N-(1-oxo-1-((pyridin-4-ylmethyl)amino)propan-2-yl)-1H-indole-2-carboxamide (RS4690), a New Dishevelled 1 InhibitorAntonio Coluccia, Marianna Bufano, Giuseppe La Regina, et al.Pageof 16