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Journal of Medicinal Chemistry
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November 19, 2019
Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere
Gwenaella Rescourio, Ana Z Gonzalez, Salman Jabri, et al.
Journal of Medicinal Chemistry
|
July 15, 2016
Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-1430)
Felix Gonzalez-Lopez de Turiso, Xiaolin Hao, Youngsook Shin, et al.
Journal of Medicinal Chemistry
|
December 4, 2014
Discovery and in vivo evaluation of (S)-N-(1-(7-fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and related PI3Kδ inhibitors for inflammation and autoimmune disease
Timothy D Cushing, Xiaolin Hao, Youngsook Shin, et al.
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Search research articles
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Showing results (11-20 of 13) with videos related to
Sort By:
Page
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You have reached the last page of results.
This site can display upto 13 results.
Journal of Medicinal Chemistry
|
November 19, 2019
Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere
Gwenaella Rescourio, Ana Z Gonzalez, Salman Jabri, et al.
Journal of Medicinal Chemistry
|
July 15, 2016
Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-1430)
Felix Gonzalez-Lopez de Turiso, Xiaolin Hao, Youngsook Shin, et al.
Journal of Medicinal Chemistry
|
December 4, 2014
Discovery and in vivo evaluation of (S)-N-(1-(7-fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine (AMG319) and related PI3Kδ inhibitors for inflammation and autoimmune disease
Timothy D Cushing, Xiaolin Hao, Youngsook Shin, et al.
Page
of 2