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Biorxiv : the Preprint Server for Biology|June 4, 2026
Ratiometric transcriptional activation by protein degradationMelissa A Gray, Katelyn L Randal, Jennifer A Co, et al.Cell Chemical Biology|May 27, 2026
The molecular basis for nuclear pore destruction by a proximity-inducing molecular glueStephen M Hinshaw, Linjie Yuan, Md Abdullah Al Noman, et al.RSC Chemical Biology|September 21, 2022
Cereblon covalent modulation through structure-based design of histidine targeting chemical probesJustin T Cruite, Geoffrey P Dann, Jianwei Che, et al.ACS Chemical Biology|May 26, 2016
Development of Chemical Probes for Investigation of Salt-Inducible Kinase Function in VivoThomas B Sundberg, Yanke Liang, Huixian Wu, et al.Nature|February 18, 2016
Inhibiting fungal multidrug resistance by disrupting an activator-Mediator interactionJoy L Nishikawa, Andras Boeszoermenyi, Luis A Vale-Silva, et al.Nature Communications|July 27, 2022
Targeting transcription in heart failure via CDK7/12/13 inhibitionAustin Hsu, Qiming Duan, Daniel S Day, et al.Molecular Cancer Therapeutics|April 15, 2018
RAS-MAPK Reactivation Facilitates Acquired Resistance in FGFR1-Amplified Lung Cancer and Underlies a Rationale for Upfront FGFR-MEK BlockadeBruno Bockorny, Maria Rusan, Wankun Chen, et al.Chembiochem : a European Journal of Chemical Biology|April 23, 2023
Development and Characterization of Selective FAK Inhibitors and PROTACs with In Vivo ActivityEriko Koide, Mikaela L Mohardt, Zainab M Doctor, et al.Nature Chemical Biology|March 28, 2018
The dTAG system for immediate and target-specific protein degradationBehnam Nabet, Justin M Roberts, Dennis L Buckley, et al.Journal of Medicinal Chemistry|April 17, 2020
Discovery and Structure-Activity Relationship Study of (Z)-5-Methylenethiazolidin-4-one Derivatives as Potent and Selective Pan-phosphatidylinositol 5-Phosphate 4-Kinase InhibitorsTheresa D Manz, Sindhu Carmen Sivakumaren, Fleur M Ferguson, et al.Pageof 156