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Journal of Medicinal Chemistry|December 4, 2009

Synthesis and in vitro opioid receptor functional antagonism of methyl-substituted analogues of (3R)-7-hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl]-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic)Juan Pablo Cueva, Tingwei Bill Cai, S Wayne Mascarella, et al.

Journal of Medicinal Chemistry|July 21, 2006

Synthesis and monoamine transporter binding properties of 2,3-cyclo analogues of 3beta-(4'-aminophenyl)-2beta-tropanemethanolF Ivy Carroll, Bruce E Blough, Xiaodong Huang, et al.

ACS Omega|August 14, 2023

Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-<i>1,6,7-d</i><sub></sub>Anita H Lewin, James P Hayes, Desong Zhong, et al.

Journal of Medicinal Chemistry|June 30, 2012

Synthesis and nicotinic acetylcholine receptor in vitro and in vivo pharmacological properties of 2'-fluoro-3'-(substituted phenyl)deschloroepibatidine analogues of 2'-fluoro-3'-(4-nitrophenyl)deschloroepibatidinePauline Ondachi, Ana Castro, Charles W Luetje, et al.

Journal of Medicinal Chemistry|December 22, 2005

N-substituted cis-4a-(3-hydroxyphenyl)-8a-methyloctahydroisoquinolines are opioid receptor pure antagonistsF Ivy Carroll, Sachin Chaudhari, James B Thomas, et al.

ACS Medicinal Chemistry Letters|April 24, 2012

Synthesis and Evaluation of Metabotropic Glutamate Receptor Subtype 5 Antagonists Based on Fenobam()Moses G Gichinga, Jeremy P Olson, Elizabeth Butala, et al.

ACS Chemical Neuroscience|August 30, 2018

Synthesis and Characterization of the Selective, Reversible PKC<sub>β</sub> Inhibitor (9 S)-9-[(Dimethylamino)methyl]-6,7,10,11-tetrahydro-9 H,18 H-5,21:12,17-dimethenodibenzo[ e,k]pyrrolo[3,4- h][1,4,13]oxadiazacyclohexadecine-18,20(19 H)-dione, Ruboxistaurin (LY333531)Anita H Lewin, Larry Brieaddy, Jeffrey R Deschamps, et al.

Journal of Medicinal Chemistry|June 3, 2008

Conformationally constrained analogues of N-(piperidinyl)-5-(4-chlorophenyl)-1-(2,4- dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide (SR141716): design, synthesis, computational analysis, and biological evaluationsYanan Zhang, Jason P Burgess, Marcus Brackeen, et al.

Journal of Medicinal Chemistry|February 18, 2010

Synthesis and biological evaluation of bupropion analogues as potential pharmacotherapies for smoking cessationF Ivy Carroll, Bruce E Blough, S Wayne Mascarella, et al.

Journal of Medicinal Chemistry|November 10, 2010

Nicotinic acetylcholine receptor efficacy and pharmacological properties of 3-(substituted phenyl)-2β-substituted tropanesF Ivy Carroll, Bruce E Blough, S Wayne Mascarella, et al.

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Showing results (11-20 of 48) with videos related to

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Journal of Medicinal Chemistry|December 4, 2009

Synthesis and in vitro opioid receptor functional antagonism of methyl-substituted analogues of (3R)-7-hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl]-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic)Juan Pablo Cueva, Tingwei Bill Cai, S Wayne Mascarella, et al.

Journal of Medicinal Chemistry|July 21, 2006

Synthesis and monoamine transporter binding properties of 2,3-cyclo analogues of 3beta-(4'-aminophenyl)-2beta-tropanemethanolF Ivy Carroll, Bruce E Blough, Xiaodong Huang, et al.

ACS Omega|August 14, 2023

Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-<i>1,6,7-d</i><sub></sub>Anita H Lewin, James P Hayes, Desong Zhong, et al.

Journal of Medicinal Chemistry|June 30, 2012

Synthesis and nicotinic acetylcholine receptor in vitro and in vivo pharmacological properties of 2'-fluoro-3'-(substituted phenyl)deschloroepibatidine analogues of 2'-fluoro-3'-(4-nitrophenyl)deschloroepibatidinePauline Ondachi, Ana Castro, Charles W Luetje, et al.

Journal of Medicinal Chemistry|December 22, 2005

N-substituted cis-4a-(3-hydroxyphenyl)-8a-methyloctahydroisoquinolines are opioid receptor pure antagonistsF Ivy Carroll, Sachin Chaudhari, James B Thomas, et al.

ACS Medicinal Chemistry Letters|April 24, 2012

Synthesis and Evaluation of Metabotropic Glutamate Receptor Subtype 5 Antagonists Based on Fenobam()Moses G Gichinga, Jeremy P Olson, Elizabeth Butala, et al.

ACS Chemical Neuroscience|August 30, 2018

Synthesis and Characterization of the Selective, Reversible PKC<sub>β</sub> Inhibitor (9 S)-9-[(Dimethylamino)methyl]-6,7,10,11-tetrahydro-9 H,18 H-5,21:12,17-dimethenodibenzo[ e,k]pyrrolo[3,4- h][1,4,13]oxadiazacyclohexadecine-18,20(19 H)-dione, Ruboxistaurin (LY333531)Anita H Lewin, Larry Brieaddy, Jeffrey R Deschamps, et al.

Journal of Medicinal Chemistry|June 3, 2008

Conformationally constrained analogues of N-(piperidinyl)-5-(4-chlorophenyl)-1-(2,4- dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide (SR141716): design, synthesis, computational analysis, and biological evaluationsYanan Zhang, Jason P Burgess, Marcus Brackeen, et al.

Journal of Medicinal Chemistry|February 18, 2010

Synthesis and biological evaluation of bupropion analogues as potential pharmacotherapies for smoking cessationF Ivy Carroll, Bruce E Blough, S Wayne Mascarella, et al.

Journal of Medicinal Chemistry|November 10, 2010

Nicotinic acetylcholine receptor efficacy and pharmacological properties of 3-(substituted phenyl)-2β-substituted tropanesF Ivy Carroll, Bruce E Blough, S Wayne Mascarella, et al.

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