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Scientific Reports|May 16, 2026
Production and characterization of gigastasin, a leech-derived inhibitor of complement and coagulation pathwaysAleksandra Blagojevic, Peter Rüthemann, Kevin Widmer, et al.Angewandte Chemie (International Ed. in English)|July 29, 2024
Strengthening an Intramolecular Non-Classical Hydrogen Bond to Get in Shape for BindingNorbert Varga, Martin Smieško, Xiaohua Jiang, et al.Iucrj|March 3, 2017
Mutation of Tyr137 of the universal <i>Escherichia coli</i> fimbrial adhesin FimH relaxes the tyrosine gate prior to mannose bindingSaid Rabbani, Eva-Maria Krammer, Goedele Roos, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|June 26, 2018
KinITC-One Method Supports both Thermodynamic and Kinetic SARs as Exemplified on FimH AntagonistsPascal Zihlmann, Marleen Silbermann, Timothy Sharpe, et al.Chemical Science|April 10, 2018
The price of flexibility - a case study on septanoses as pyranose mimeticsChristoph P Sager, Brigitte Fiege, Pascal Zihlmann, et al.Acta Biomaterialia|November 3, 2022
Complement-regulatory biomaterial coatings: Activity and selectivity profile of the factor H-binding peptide 5C6Clément Bechtler, Sophia Koutsogiannaki, Ekaterina Umnyakova, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|January 4, 2012
Pre-organization of the core structure of E-selectin antagonistsDaniel Schwizer, John T Patton, Brian Cutting, et al.Journal of Medicinal Chemistry|January 26, 2010
Low molecular weight antagonists of the myelin-associated glycoprotein: synthesis, docking, and biological evaluationStefanie Mesch, Delia Moser, Daniel S Strasser, et al.Journal of the American Chemical Society|October 15, 2021
Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2Jonathan Cramer, Adem Lakkaichi, Butrint Aliu, et al.Chemmedchem|February 3, 2019
Improvement of Aglycone π-Stacking Yields Nanomolar to Sub-nanomolar FimH AntagonistsWojciech Schönemann, Jonathan Cramer, Tobias Mühlethaler, et al.Pageof 5