Showing results (41-50 of 79) with videos related to
Sort By:
Pageof 8
Chemmedchem|September 30, 2017
Mimicking Intermolecular Interactions of Tight Protein-Protein Complexes for Small-Molecule AntagonistsDavid Xu, Khuchtumur Bum-Erdene, Yubing Si, et al.Chemistry & Biology|February 24, 2006
Interactions of designer antibiotics and the bacterial ribosomal aminoacyl-tRNA siteJames B Murray, Samy O Meroueh, Rupert J M Russell, et al.The Journal of Organic Chemistry|July 2, 2005
Design, synthesis, and evaluation of a mechanism-based inhibitor for gelatinase AMasahiro Ikejiri, M Margarida Bernardo, Samy O Meroueh, et al.Chemmedchem|October 27, 2020
Small-Molecule Inhibition of the uPAR ⋅ uPA Interaction by Conformational SelectionDavid Xu, Khuchtumur Bum-Erdene, Julie M Leth, et al.Proceedings of the National Academy of Sciences of the United States of America|March 18, 2020
Small-molecule covalent bond formation at tyrosine creates a binding site and inhibits activation of Ral GTPasesKhuchtumur Bum-Erdene, Degang Liu, Giovanni Gonzalez-Gutierrez, et al.Journal of Chemical Information and Modeling|March 29, 2011
Target-specific support vector machine scoring in structure-based virtual screening: computational validation, in vitro testing in kinases, and effects on lung cancer cell proliferationLiwei Li, May Khanna, Inha Jo, et al.Biochemistry|March 3, 2004
Fluorinated aminoglycosides and their mechanistic implication for aminoglycoside 3'-phosphotransferases from Gram-negative bacteriaChoonkeun Kim, Jalal Haddad, Sergei B Vakulenko, et al.Chemistry & Biology|April 25, 2006
Design and characterization of a metalloproteinase inhibitor-tethered resin for the detection of active MMPs in biological samplesDusan Hesek, Marta Toth, Samy O Meroueh, et al.Journal of Medicinal Chemistry|December 23, 2022
Small-Molecule Cyanamide Pan-TEAD·YAP1 Covalent AntagonistsKhuchtumur Bum-Erdene, I-Ju Yeh, Giovanni Gonzalez-Gutierrez, et al.Bioorganic & Medicinal Chemistry|April 26, 2017
Small molecules inhibit STAT3 activation, autophagy, and cancer cell anchorage-independent growthDonghui Zhou, Maya Z Springer, David Xu, et al.Pageof 8