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Chemmedchem|September 18, 2018
Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1H)-one Scaffold Using Palladium-Catalysed Cross-Coupling ReactionsJulien Pedron, Clotilde Boudot, Sandra Bourgeade-Delmas, et al.Pharmaceuticals (Basel, Switzerland)|August 26, 2022
Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo[1,2-a]pyridine Antileishmanial PharmacophoreRomain Paoli-Lombardo, Nicolas Primas, Sandra Bourgeade-Delmas, et al.Chemistry (Weinheim an Der Bergstrasse, Germany)|July 10, 2026
Fluorine Makes the Difference-Gold(I)-NHC Complexes With Fluoroaryl Substituents Exhibit Highly Potent Antileishmanial ActivitySoumia Ftouh, Sandra Bourgeade-Delmas, Chloé Salis, et al.European Journal of Medicinal Chemistry|June 10, 2018
Novel 8-nitroquinolin-2(1H)-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR studyJulien Pedron, Clotilde Boudot, Sébastien Hutter, et al.Journal of Lipid Research|January 11, 2019
Polyunsaturated fatty acid metabolites: biosynthesis in Leishmania and role in parasite/host interactionLucie Paloque, Teresa Perez-Berezo, Anne Abot, et al.European Journal of Medicinal Chemistry|August 10, 2018
8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductasesCyril Fersing, Clotilde Boudot, Julien Pedron, et al.ACS Medicinal Chemistry Letters|January 19, 2019
Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial ActivityCyril Fersing, Louise Basmaciyan, Clotilde Boudot, et al.ACS Medicinal Chemistry Letters|April 16, 2020
New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruziJulien Pedron, Clotilde Boudot, Jean-Yves Brossas, et al.European Journal of Medicinal Chemistry|August 16, 2020
Antikinetoplastid SAR study in 3-nitroimidazopyridine series: Identification of a novel non-genotoxic and potent anti-T. b. brucei hit-compound with improved pharmacokinetic propertiesCyril Fersing, Clotilde Boudot, Romain Paoli-Lombardo, et al.European Journal of Medicinal Chemistry|July 12, 2020
8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruziCyril Fersing, Clotilde Boudot, Caroline Castera-Ducros, et al.Pageof 3