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Food & Function|May 29, 2019
Dietary polyphenols rutin, taxifolin and quercetin related compounds target Leishmania amazonensis arginaseEdson Roberto da Silva, Simone Brogi, João Francisco Lucon-Júnior, et al.Journal of Natural Products|April 21, 2016
Verbascoside Inhibits Promastigote Growth and Arginase Activity of Leishmania amazonensisClaudia C Maquiaveli, João F Lucon-Júnior, Simone Brogi, et al.Chemical Biology & Drug Design|September 15, 2018
Cinnamic acids derived compounds with antileishmanial activity target Leishmania amazonensis arginaseEdson Roberto da Silva, Simone Brogi, Alessandro Grillo, et al.Antimicrobial Agents and Chemotherapy|April 24, 2004
Effects of drug resistance mutations L100I and V106A on the binding of pyrrolobenzoxazepinone nonnucleoside inhibitors to the human immunodeficiency virus type 1 reverse transcriptase catalytic complexGiada A Locatelli, Giuseppe Campiani, Reynel Cancio, et al.The Journal of Biological Chemistry|September 15, 2011
The Ca2+-ATPase (SERCA1) is inhibited by 4-aminoquinoline derivatives through interference with catalytic activation by Ca2+, whereas the ATPase E2 state remains functionalGianluca Bartolommei, Francesco Tadini-Buoninsegni, Maria Rosa Moncelli, et al.Journal of Medicinal Chemistry|September 12, 2008
Flexible cyclic ethers/polyethers as novel P2-ligands for HIV-1 protease inhibitors: design, synthesis, biological evaluation, and protein-ligand X-ray studiesArun K Ghosh, Sandra Gemma, Abigail Baldridge, et al.Pathogens (Basel, Switzerland)|September 23, 2022
In Vitro and In Silico Analyses of New Cinnamid and Rosmarinic Acid-Derived Compounds Biosynthesized in <i>Escherichia coli</i> as <i>Leishmania amazonensis</i> Arginase InhibitorsJulio Abel Alfredo Dos Santos Simone Come, Yibin Zhuang, Tianzhen Li, et al.Bioorganic & Medicinal Chemistry Letters|June 10, 2014
Rational design of the first difluorostatone-based PfSUB1 inhibitorsSimone Giovani, Maria Penzo, Simone Brogi, et al.Molecules (Basel, Switzerland)|September 28, 2023
Development of Quinazolinone Derivatives as Modulators of Virulence Factors of <i>Pseudomonas aeruginosa</i> Cystic Fibrosis StrainsGabriele Carullo, Giovanni Di Bonaventura, Sara Rossi, et al.Chemical Biology & Drug Design|January 17, 2024
Synthetic derivatives of natural cinnamic acids as potential anti-colorectal cancer agentsFederica Falbo, Sandra Gemma, Adrian Koch, et al.Pageof 15