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The Journal of Biological Chemistry|August 15, 2022
Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitorsFulvio Saccoccia, Luca Pozzetti, Roberto Gimmelli, et al.Chemmedchem|November 14, 2017
Activation of the Wnt Pathway by Small Peptides: Rational Design, Synthesis and Biological EvaluationSimone Brogi, Samuele Maramai, Margherita Brindisi, et al.Chemical Biology & Drug Design|August 6, 2015
Site-directed Mutagenesis of Key Residues Unveiled a Novel Allosteric Site on Human Adenosine Kinase for Pyrrolobenzoxa(thia)zepinone Non-Nucleoside InhibitorsLida Savi, Margherita Brindisi, Gloria Alfano, et al.Bioorganic & Medicinal Chemistry Letters|July 17, 2012
Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1Sandra Gemma, Simone Giovani, Margherita Brindisi, et al.Bioorganic & Medicinal Chemistry Letters|October 1, 2010
Discovery of potent nucleotide-mimicking competitive inhibitors of hepatitis C virus NS3 helicaseSandra Gemma, Stefania Butini, Giuseppe Campiani, et al.Journal of Medicinal Chemistry|July 19, 2011
Synthesis and antiplasmodial activity of bicyclic dioxanes as simplified dihydroplakortin analoguesSandra Gemma, Sanil Kunjir, Salvatore Sanna Coccone, et al.ACS Chemical Neuroscience|May 22, 2020
Ionotropic Glutamate Receptor GluA2 in Complex with Bicyclic Pyrimidinedione-Based Compounds: When Small Compound Modifications Have Distinct Effects on Binding InteractionsKarla Frydenvang, Darryl S Pickering, Giridhar U Kshirsagar, et al.Archiv Der Pharmazie|September 26, 2023
Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agentsAlessandro Papa, Ilaria Cursaro, Luca Pozzetti, et al.The Journal of Organic Chemistry|October 11, 2008
An efficient approach to chiral C8/C9-piperazino-substituted 1,4-benzodiazepin-2-ones as peptidomimetic scaffoldsStefania Butini, Emanuele Gabellieri, Paul Brady Huleatt, et al.Journal of Medicinal Chemistry|May 26, 2006
Discovery of huperzine A-tacrine hybrids as potent inhibitors of human cholinesterases targeting their midgorge recognition sitesSandra Gemma, Emanuele Gabellieri, Paul Huleatt, et al.Pageof 15