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ACS Medicinal Chemistry Letters|May 14, 2025
Discovery of <i>p</i>-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox VirusSara Rossi, Luca Pozzetti, Gabriele Carullo, et al.Journal of Food Science|November 14, 2023
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessmentRiccardo Fedeli, Ludovica Marotta, Luca Frattaruolo, et al.Bioorganic & Medicinal Chemistry Letters|August 8, 2006
Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strainsSandra Gemma, Gagan Kukreja, Caterina Fattorusso, et al.Biochemical Pharmacology|June 11, 2008
Selective targeting of the HIV-1 reverse transcriptase catalytic complex through interaction with the "primer grip" region by pyrrolobenzoxazepinone non-nucleoside inhibitors correlates with increased activity towards drug-resistant mutantsSamantha Zanoli, Sandra Gemma, Stefania Butini, et al.Scientific Reports|May 8, 2015
Structure-based discovery of the first non-covalent inhibitors of Leishmania major tryparedoxin peroxidase by high throughput dockingMargherita Brindisi, Simone Brogi, Nicola Relitti, et al.Bioorganic & Medicinal Chemistry|July 22, 2009
Development of antitubercular compounds based on a 4-quinolylhydrazone scaffold. Further structure-activity relationship studiesSandra Gemma, Luisa Savini, Maria Altarelli, et al.Chemmedchem|October 4, 2022
Synthesis of Unsymmetrical Squaramides as Allosteric GSK-3β Inhibitors Promoting β-Catenin-Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial CellsGabriele Carullo, Laura Bottoni, Silvia Pasquini, et al.Organic & Biomolecular Chemistry|October 10, 2008
Potent HIV-1 protease inhibitors incorporating meso-bicyclic urethanes as P2-ligands: structure-based design, synthesis, biological evaluation and protein-ligand X-ray studiesArun K Ghosh, Sandra Gemma, Jun Takayama, et al.Bioorganic & Medicinal Chemistry Letters|June 4, 2011
Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutantsStefania Butini, Sandra Gemma, Margherita Brindisi, et al.Bioorganic & Medicinal Chemistry Letters|December 15, 2012
Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition propertiesStefania Butini, Sandra Gemma, Margherita Brindisi, et al.Pageof 15