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Sandrine Ruchaud

Showing results (51-60 of 65) with videos related to

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Scientific Reports|April 18, 2025
Development of a novel family of antifungal agents based on a quinone methide oxime frameworkMonika Janeczko, Maciej Masłyk, Oleg M Demchuk, et al.
European Journal of Medicinal Chemistry|March 29, 2016
Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitorsAziz Ouach, Rajâa Boulahjar, Christine Vala, et al.
European Journal of Medicinal Chemistry|October 16, 2012
Synthesis and biological evaluation of new 5-benzylated 4-oxo-3,4-dihydro-5H-pyridazino[4,5-b]indoles as PI3Kα inhibitorsAmélie Bruel, Cédric Logé, Marie-Ludivine de Tauzia, et al.
Antimicrobial Agents and Chemotherapy|February 24, 2016
From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial ActivityEmilie Durieu, Eric Prina, Olivier Leclercq, et al.
European Journal of Medicinal Chemistry|September 19, 2015
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazinesPascal Marchand, Marc-Antoine Bazin, Fabrice Pagniez, et al.
Molecules (Basel, Switzerland)|November 16, 2018
From Quinoxaline, Pyrido[2,3-<i>b</i>]pyrazine and Pyrido[3,4-<i>b</i>]pyrazine to Pyrazino-Fused Carbazoles and CarbolinesFrédéric Lassagne, Timothy Langlais, Elsa Caytan, et al.
Anti-Cancer Agents in Medicinal Chemistry|December 9, 2016
Discovery of New Aminosubstituted Pyrrolopyrimidines with Antiproliferative Activity Against Breast Cancer Cells and Investigation of their Effect Towards the PI3Kα EnzymeKonstantinos Daniilides, Nikolaos Lougiakis, Thomas Evangelidis, et al.
Bioorganic & Medicinal Chemistry|January 10, 2021
Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinaseDabbugoddu Brahmaiah, Anagani Kanaka Durga Bhavani, Pasula Aparna, et al.
Molecules (Basel, Switzerland)|October 14, 2022
Structure Activity Relationship Studies around <i>DB18</i>, a Potent and Selective Inhibitor of CLK KinasesDabbugoddu Brahmaiah, Anagani Kanaka Durga Bhavani, Pasula Aparna, et al.
The Journal of Biological Chemistry|October 26, 2001
Lack of correlation between caspase activation and caspase activity assays in paclitaxel-treated MCF-7 breast cancer cellsTimothy J Kottke, April L Blajeski, X Wei Meng, et al.
Pageof 7

Showing results (51-60 of 65) with videos related to

Sort By:
Pageof 7
Scientific Reports|April 18, 2025
Development of a novel family of antifungal agents based on a quinone methide oxime frameworkMonika Janeczko, Maciej Masłyk, Oleg M Demchuk, et al.
European Journal of Medicinal Chemistry|March 29, 2016
Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitorsAziz Ouach, Rajâa Boulahjar, Christine Vala, et al.
European Journal of Medicinal Chemistry|October 16, 2012
Synthesis and biological evaluation of new 5-benzylated 4-oxo-3,4-dihydro-5H-pyridazino[4,5-b]indoles as PI3Kα inhibitorsAmélie Bruel, Cédric Logé, Marie-Ludivine de Tauzia, et al.
Antimicrobial Agents and Chemotherapy|February 24, 2016
From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial ActivityEmilie Durieu, Eric Prina, Olivier Leclercq, et al.
European Journal of Medicinal Chemistry|September 19, 2015
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazinesPascal Marchand, Marc-Antoine Bazin, Fabrice Pagniez, et al.
Molecules (Basel, Switzerland)|November 16, 2018
From Quinoxaline, Pyrido[2,3-<i>b</i>]pyrazine and Pyrido[3,4-<i>b</i>]pyrazine to Pyrazino-Fused Carbazoles and CarbolinesFrédéric Lassagne, Timothy Langlais, Elsa Caytan, et al.
Anti-Cancer Agents in Medicinal Chemistry|December 9, 2016
Discovery of New Aminosubstituted Pyrrolopyrimidines with Antiproliferative Activity Against Breast Cancer Cells and Investigation of their Effect Towards the PI3Kα EnzymeKonstantinos Daniilides, Nikolaos Lougiakis, Thomas Evangelidis, et al.
Bioorganic & Medicinal Chemistry|January 10, 2021
Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinaseDabbugoddu Brahmaiah, Anagani Kanaka Durga Bhavani, Pasula Aparna, et al.
Molecules (Basel, Switzerland)|October 14, 2022
Structure Activity Relationship Studies around <i>DB18</i>, a Potent and Selective Inhibitor of CLK KinasesDabbugoddu Brahmaiah, Anagani Kanaka Durga Bhavani, Pasula Aparna, et al.
The Journal of Biological Chemistry|October 26, 2001
Lack of correlation between caspase activation and caspase activity assays in paclitaxel-treated MCF-7 breast cancer cellsTimothy J Kottke, April L Blajeski, X Wei Meng, et al.
Pageof 7