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Molecules (Basel, Switzerland)|March 27, 2025
Design, Synthesis, and Biological Evaluation of 5,8-Dimethyl Shikonin Oximes as SARS-CoV-2 Mpro InhibitorsJiahua Cui, Shouyan Xiang, Qijing Zhang, et al.RSC Advances|May 11, 2022
Development of 2-arylbenzo[h]quinolone analogs as selective CYP1B1 inhibitorsJinyun Dong, Zengtao Wang, Qingqing Meng, et al.Journal of Medicinal Chemistry|November 30, 2023
Design and Synthesis of Novel Near-Infrared Fluorescence Probes Based on an Open Conformation of a Cytochrome P450 1B1 Complex for Molecular Imaging of Colorectal TumorsDongmei Chen, Ruining Li, Qi Shao, et al.Molecular Pharmaceutics|November 28, 2018
DMAKO-20 as a New Multitarget Anticancer Prodrug Activated by the Tumor Specific CYP1B1 EnzymeJiahua Cui, Xu Zhang, Guang Huang, et al.Medchemcomm|December 6, 2019
Development of benzochalcone derivatives as selective CYP1B1 inhibitors and anticancer agentsJinyun Dong, Guang Huang, Qijing Zhang, et al.Cancer Letters|December 14, 2011
Cryptotanshinone suppresses androgen receptor-mediated growth in androgen dependent and castration resistant prostate cancer cellsDefeng Xu, Tzu-Hua Lin, Shaoshun Li, et al.Anti-Cancer Agents in Medicinal Chemistry|April 6, 2021
Design, Synthesis and Binding Affinity Evaluation of Cytochrome P450 1B1 Targeted ChelatorsDongmei Chen, Qiqi Fan, Ting Xu, et al.Journal of Medicinal Chemistry|June 5, 2023
Discovery of Dimethyl Shikonin Oxime 5a, a Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Type 2 Diabetes MellitusLehao Wu, Jiahua Cui, Chunxiao Zhao, et al.Molecular Pharmaceutics|January 31, 2025
Application of a CYP1B1-Targeted NIR Probe for Breast Cancer Diagnosis, Surgical Navigation, and CYP1B1-Associated Chemotherapy Resistance MonitoringZhihao Wu, Tao Shi, Qi Shao, et al.Chembiochem : a European Journal of Chemical Biology|May 14, 2022
Design, Synthesis and In Vivo Fluorescence Imaging Study of a Cytochrome P450 1B1 Targeted NIR Probe Containing a Chelator MoietyZengtao Wang, Dongmei Chen, Qiqi Fan, et al.Pageof 4