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Journal of Medicinal Chemistry|June 23, 2009
Identification of an orally active opioid receptor-like 1 (ORL1) receptor antagonist 4-{3-[(2R)-2,3-dihydroxypropyl]-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl}-1-[(1S,3S,4R)-spiro[bicyclo[2.2.1]heptane-2,1'-cyclopropan]-3-ylmethyl]piperidine as clinical candidateAtsushi Satoh, Takeshi Sagara, Hiroki Sakoh, et al.Bioorganic & Medicinal Chemistry|April 27, 2016
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibitionHideyuki Igawa, Masashi Takahashi, Mikio Shirasaki, et al.Journal of Medicinal Chemistry|June 10, 2008
A novel class of cycloalkano[b]pyridines as potent and orally active opioid receptor-like 1 antagonists with minimal binding affinity to the hERG K+ channelTakashi Yoshizumi, Hirobumi Takahashi, Hiroshi Miyazoe, et al.Pageof 3