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Journal of Medicinal Chemistry
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December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma
Cristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
European Journal of Medicinal Chemistry
|
November 8, 2012
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme
Mariangela Biava, Claudio Battilocchio, Giovanna Poce, et al.
Cellular Physiology and Biochemistry : International Journal of Experimental Cellular Physiology, Biochemistry, and Pharmacology
|
April 15, 2015
SI113, a specific inhibitor of the Sgk1 kinase activity that counteracts cancer cell proliferation
Lucia D'Antona, Rosario Amato, Cristina Talarico, et al.
Bioorganic Chemistry
|
August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment
Salvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
Oncotarget
|
August 28, 2016
A Pyrazolo[3,4-d]pyrimidine compound inhibits Fyn phosphorylation and induces apoptosis in natural killer cell leukemia
Ilaria Laurenzana, Antonella Caivano, Stefania Trino, et al.
Journal of Medicinal Chemistry
|
June 27, 2017
Prodrugs of Pyrazolo[3,4-d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model
Giulia Vignaroli, Giulia Iovenitti, Claudio Zamperini, et al.
International Journal of Molecular Sciences
|
September 27, 2019
Proton Therapy and Src Family Kinase Inhibitor Combined Treatments on U87 Human Glioblastoma Multiforme Cell Line
Francesco P Cammarata, Filippo Torrisi, Giusi I Forte, et al.
Journal of Medicinal Chemistry
|
May 27, 2005
Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives
Angelo Ranise, Andrea Spallarossa, Sara Cesarini, et al.
Journal of Medicinal Chemistry
|
October 13, 2007
Identification of a novel pyrazolo[3,4-d]pyrimidine able to inhibit cell proliferation of a human osteogenic sarcoma in vitro and in a xenograft model in mice
Fabrizio Manetti, Annalisa Santucci, Giada A Locatelli, et al.
Cancers
|
June 29, 2019
A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4-<i>d</i>]Pyrimidine Dual Src/P-Glycoprotein Inhibitor
Anna Lucia Fallacara, Claudio Zamperini, Ana Podolski-Renić, et al.
Page
of 18
Search research articles
Search
Showing results (161-170 of 173) with videos related to
Sort By:
Page
of 18
Journal of Medicinal Chemistry
|
December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma
Cristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
European Journal of Medicinal Chemistry
|
November 8, 2012
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme
Mariangela Biava, Claudio Battilocchio, Giovanna Poce, et al.
Cellular Physiology and Biochemistry : International Journal of Experimental Cellular Physiology, Biochemistry, and Pharmacology
|
April 15, 2015
SI113, a specific inhibitor of the Sgk1 kinase activity that counteracts cancer cell proliferation
Lucia D'Antona, Rosario Amato, Cristina Talarico, et al.
Bioorganic Chemistry
|
August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment
Salvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
Oncotarget
|
August 28, 2016
A Pyrazolo[3,4-d]pyrimidine compound inhibits Fyn phosphorylation and induces apoptosis in natural killer cell leukemia
Ilaria Laurenzana, Antonella Caivano, Stefania Trino, et al.
Journal of Medicinal Chemistry
|
June 27, 2017
Prodrugs of Pyrazolo[3,4-d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model
Giulia Vignaroli, Giulia Iovenitti, Claudio Zamperini, et al.
International Journal of Molecular Sciences
|
September 27, 2019
Proton Therapy and Src Family Kinase Inhibitor Combined Treatments on U87 Human Glioblastoma Multiforme Cell Line
Francesco P Cammarata, Filippo Torrisi, Giusi I Forte, et al.
Journal of Medicinal Chemistry
|
May 27, 2005
Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives
Angelo Ranise, Andrea Spallarossa, Sara Cesarini, et al.
Journal of Medicinal Chemistry
|
October 13, 2007
Identification of a novel pyrazolo[3,4-d]pyrimidine able to inhibit cell proliferation of a human osteogenic sarcoma in vitro and in a xenograft model in mice
Fabrizio Manetti, Annalisa Santucci, Giada A Locatelli, et al.
Cancers
|
June 29, 2019
A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4-<i>d</i>]Pyrimidine Dual Src/P-Glycoprotein Inhibitor
Anna Lucia Fallacara, Claudio Zamperini, Ana Podolski-Renić, et al.
Page
of 18