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Drug Metabolism and Pharmacokinetics
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May 23, 2014
CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction
Claudio Zamperini, Elena Dreassi, Giulia Vignaroli, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 1, 2017
Pyrazolo[3,4-d]pyrimidines-loaded human serum albumin (HSA) nanoparticles: Preparation, characterization and cytotoxicity evaluation against neuroblastoma cell line
Anna Lucia Fallacara, Arianna Mancini, Claudio Zamperini, et al.
European Journal of Medicinal Chemistry
|
October 29, 2008
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
Andrea Spallarossa, Sara Cesarini, Angelo Ranise, et al.
Molecules (Basel, Switzerland)
|
April 27, 2024
Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling
Giancarlo Grossi, Naomi Scarano, Francesca Musumeci, et al.
European Journal of Medicinal Chemistry
|
October 26, 2010
2-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors
Elena Dreassi, Alessandra Tania Zizzari, Mattia Mori, et al.
Organic & Biomolecular Chemistry
|
July 13, 2005
New pyrazolo[3,4-b]pyridones as selective A(1) adenosine receptor antagonists: synthesis, biological evaluation and molecular modelling studies
Paola Fossa, Marco Pestarino, Giulia Menozzi, et al.
Bioorganic & Medicinal Chemistry
|
May 27, 2008
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
Sara Cesarini, Andrea Spallarossa, Angelo Ranise, et al.
Chemmedchem
|
February 14, 2007
Inhibition of Bcr-Abl phosphorylation and induction of apoptosis by pyrazolo[3,4-d]pyrimidines in human leukemia cells
Fabrizio Manetti, Annalisa Pucci, Matteo Magnani, et al.
Journal of Medicinal Chemistry
|
February 21, 2003
Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: a novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives
Angelo Ranise, Andrea Spallarossa, Silvia Schenone, et al.
Future Medicinal Chemistry
|
December 16, 2014
The search for a common structural moiety among selected pharmacological correctors of the mutant CFTR chloride channel
Erika Nieddu, Benedetta Pollarolo, Marco T Mazzei, et al.
Page
of 18
Search research articles
Search
Showing results (71-80 of 173) with videos related to
Sort By:
Page
of 18
Drug Metabolism and Pharmacokinetics
|
May 23, 2014
CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction
Claudio Zamperini, Elena Dreassi, Giulia Vignaroli, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 1, 2017
Pyrazolo[3,4-d]pyrimidines-loaded human serum albumin (HSA) nanoparticles: Preparation, characterization and cytotoxicity evaluation against neuroblastoma cell line
Anna Lucia Fallacara, Arianna Mancini, Claudio Zamperini, et al.
European Journal of Medicinal Chemistry
|
October 29, 2008
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
Andrea Spallarossa, Sara Cesarini, Angelo Ranise, et al.
Molecules (Basel, Switzerland)
|
April 27, 2024
Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling
Giancarlo Grossi, Naomi Scarano, Francesca Musumeci, et al.
European Journal of Medicinal Chemistry
|
October 26, 2010
2-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors
Elena Dreassi, Alessandra Tania Zizzari, Mattia Mori, et al.
Organic & Biomolecular Chemistry
|
July 13, 2005
New pyrazolo[3,4-b]pyridones as selective A(1) adenosine receptor antagonists: synthesis, biological evaluation and molecular modelling studies
Paola Fossa, Marco Pestarino, Giulia Menozzi, et al.
Bioorganic & Medicinal Chemistry
|
May 27, 2008
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
Sara Cesarini, Andrea Spallarossa, Angelo Ranise, et al.
Chemmedchem
|
February 14, 2007
Inhibition of Bcr-Abl phosphorylation and induction of apoptosis by pyrazolo[3,4-d]pyrimidines in human leukemia cells
Fabrizio Manetti, Annalisa Pucci, Matteo Magnani, et al.
Journal of Medicinal Chemistry
|
February 21, 2003
Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: a novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives
Angelo Ranise, Andrea Spallarossa, Silvia Schenone, et al.
Future Medicinal Chemistry
|
December 16, 2014
The search for a common structural moiety among selected pharmacological correctors of the mutant CFTR chloride channel
Erika Nieddu, Benedetta Pollarolo, Marco T Mazzei, et al.
Page
of 18