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The Journal of Organic Chemistry|November 20, 2015
Synthesis of 4-Arylthieno[2,3-b]pyridines and 4-Aminothieno[2,3-b]pyridines via a Regioselective Bromination of Thieno[2,3-b]pyridineSimon C C Lucas, Jane E Moore, Craig S Donald, et al.SLAS Discovery : Advancing Life Sciences R & D|January 26, 2024
Covalent hits and where to find themSimon C C Lucas, J Henry Blackwell, Sarah H Hewitt, et al.Drug Discovery Today|August 22, 2024
Hit me with your best shot: Integrated hit discovery for the next generation of drug targetsS Neha Ashraf, J Henry Blackwell, Geoffrey A Holdgate, et al.RSC Medicinal Chemistry|May 3, 2021
Put a ring on it: application of small aliphatic rings in medicinal chemistryMatthias R Bauer, Paolo Di Fruscia, Simon C C Lucas, et al.The Journal of Organic Chemistry|May 30, 2018
Alkene Oxyamination Using Malonoyl Peroxides: Preparation of Pyrrolidines and IsoxazolidinesCarla Alamillo-Ferrer, Jonathan M Curle, Stuart C Davidson, et al.ACS Medicinal Chemistry Letters|April 16, 2025
Discovery of a Series of Covalent Ligands That Bind to Cys77 of the Von Hippel-Lindau Tumor Suppressor Protein (VHL)Simon C C Lucas, Yong Xu, Sarah Hewitt, et al.Journal of the American Chemical Society|July 30, 2025
Modular Synthetic Platform for the Elaboration of Fragments in Three Dimensions for Fragment-Based Drug DiscoveryAndres R Gomez-Angel, Hanna F Klein, Stephen Y Yao, et al.Journal of Medicinal Chemistry|April 24, 2020
Optimization of Potent ATAD2 and CECR2 Bromodomain Inhibitors with an Atypical Binding ModeSimon C C Lucas, Stephen J Atkinson, Paul Bamborough, et al.RSC Medicinal Chemistry|November 3, 2022
Fragment screening at AstraZeneca: developing the next generation biophysics fragment setSimon C C Lucas, Ulf Börjesson, Mark J Bostock, et al.ACS Medicinal Chemistry Letters|June 18, 2025
Discovery of Pyrimidoindolones as Novel Family VIII Bromodomain BindersJeffrey A Boerth, Marianne Schimpl, Simon C C Lucas, et al.Pageof 3