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European Journal of Medicinal Chemistry
|
May 22, 2022
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models
Veronica Di Sarno, Pia Giovannelli, Alicia Medina-Peris, et al.
Journal of Medicinal Chemistry
|
June 26, 2018
Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity
Alessia Bertamino, Nunzio Iraci, Carmine Ostacolo, et al.
Chemmedchem
|
May 6, 2025
Novel Para-Phenylenediamine-Based Derivatives as Receptor Tyrosine Kinase-like Orphan Receptor 1 (ROR1) Inhibitors: An In Vitro Preliminary Characterization
Gerardina Smaldone, Maria Rosaria Miranda, Francesca Di Matteo, et al.
Journal of Medicinal Chemistry
|
August 16, 2022
Beyond Retigabine: Design, Synthesis, and Pharmacological Characterization of a Potent and Chemically Stable Neuronal Kv7 Channel Activator with Anticonvulsant Activity
Simona Musella, Lidia Carotenuto, Nunzio Iraci, et al.
European Journal of Medicinal Chemistry
|
September 27, 2021
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization
Veronica Di Sarno, Gianluigi Lauro, Simona Musella, et al.
Journal of Medicinal Chemistry
|
December 10, 2019
Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel Activators
Carmine Ostacolo, Francesco Miceli, Veronica Di Sarno, et al.
ACS Chemical Biology
|
May 1, 2013
Discovery of PTPRJ agonist peptides that effectively inhibit in vitro cancer cell proliferation and tube formation
Francesco Ortuso, Francesco Paduano, Alfonso Carotenuto, et al.
European Journal of Medicinal Chemistry
|
January 17, 2024
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization
Tania Ciaglia, Vincenzo Vestuto, Veronica Di Sarno, et al.
Journal of Medicinal Chemistry
|
July 24, 2025
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution
Tania Ciaglia, Valeria Napolitano, Maria Rosaria Miranda, et al.
Journal of Medicinal Chemistry
|
June 19, 2023
Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis
Simona Musella, Danilo D'Avino, Lukas Klaus Peltner, et al.
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Search research articles
Search
Showing results (41-50 of 55) with videos related to
Sort By:
Page
of 6
European Journal of Medicinal Chemistry
|
May 22, 2022
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models
Veronica Di Sarno, Pia Giovannelli, Alicia Medina-Peris, et al.
Journal of Medicinal Chemistry
|
June 26, 2018
Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity
Alessia Bertamino, Nunzio Iraci, Carmine Ostacolo, et al.
Chemmedchem
|
May 6, 2025
Novel Para-Phenylenediamine-Based Derivatives as Receptor Tyrosine Kinase-like Orphan Receptor 1 (ROR1) Inhibitors: An In Vitro Preliminary Characterization
Gerardina Smaldone, Maria Rosaria Miranda, Francesca Di Matteo, et al.
Journal of Medicinal Chemistry
|
August 16, 2022
Beyond Retigabine: Design, Synthesis, and Pharmacological Characterization of a Potent and Chemically Stable Neuronal Kv7 Channel Activator with Anticonvulsant Activity
Simona Musella, Lidia Carotenuto, Nunzio Iraci, et al.
European Journal of Medicinal Chemistry
|
September 27, 2021
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization
Veronica Di Sarno, Gianluigi Lauro, Simona Musella, et al.
Journal of Medicinal Chemistry
|
December 10, 2019
Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel Activators
Carmine Ostacolo, Francesco Miceli, Veronica Di Sarno, et al.
ACS Chemical Biology
|
May 1, 2013
Discovery of PTPRJ agonist peptides that effectively inhibit in vitro cancer cell proliferation and tube formation
Francesco Ortuso, Francesco Paduano, Alfonso Carotenuto, et al.
European Journal of Medicinal Chemistry
|
January 17, 2024
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization
Tania Ciaglia, Vincenzo Vestuto, Veronica Di Sarno, et al.
Journal of Medicinal Chemistry
|
July 24, 2025
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution
Tania Ciaglia, Valeria Napolitano, Maria Rosaria Miranda, et al.
Journal of Medicinal Chemistry
|
June 19, 2023
Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis
Simona Musella, Danilo D'Avino, Lukas Klaus Peltner, et al.
Page
of 6