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Journal of Enzyme Inhibition and Medicinal Chemistry|November 23, 2023
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamatesSimone Giovannuzzi, Anil Kumar Marapaka, Nader S Abutaleb, et al.
European Journal of Medicinal Chemistry|April 23, 2025
Redesigning oxazolidinones as carbonic anhydrase inhibitors against vancomycin-resistant enterococciAndrea Ammara, Simone Giovannuzzi, Alessandro Bonardi, et al.
International Journal of Biological Macromolecules|January 30, 2025
Development of pyrazolo[1,5-a]pyrimidine-grafted coumarins as selective carbonic anhydrase inhibitors and tubulin polymerization inhibitors with potent anticancer activityMahmoud S Elkotamy, Mohamed A Abdelrahman, Simone Giovannuzzi, et al.
European Journal of Medicinal Chemistry|March 29, 2026
Multi-target pyrazolopyrimidine-coumarin derivatives as potent CA IX/XII and tubulin polymerization inhibitors: Design, synthesis, and biological evaluationMahmoud S Elkotamy, Mohamed A Abdelrahman, Simone Giovannuzzi, et al.
Journal of Medicinal Chemistry|January 26, 2026
First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic AgentsEslam Roshdy, Eva Řezníčková, Mostafa M Elbadawi, et al.
Journal of Medicinal Chemistry|July 28, 2023
1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory ActivitiesAhmed E Elsawi, Mostafa M Elbadawi, Alessio Nocentini, et al.
Archiv Der Pharmazie|December 23, 2024
Depsides from Origanum dictamnus and Satureja pilosa as selective inhibitors of carbonic anhydrases: Isolation, structure elucidation, X-ray crystallographyCharikleia Paloukopoulou, Ogouschan Salim Ntagli, Luca Gherardi, et al.
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