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The AAPS Journal|September 4, 2023
Human Brain Penetration Prediction Using Scaling Approach from Animal Machine Learning ModelsSiyu Liu, Yohei KosugiMolecular Pharmaceutics|January 29, 2021
Prediction of Oral Pharmacokinetics Using a Combination of In Silico Descriptors and In Vitro ADME PropertiesYohei Kosugi, Natalie HoseaXenobiotica; the Fate of Foreign Compounds in Biological Systems|November 12, 2014
Species differences and substrate specificity of CYP3A heteroactivation by efavirenzYohei Kosugi, Junzo TakahashiMolecular Pharmaceutics|June 2, 2020
Direct Comparison of Total Clearance Prediction: Computational Machine Learning Model versus Bottom-Up Approach Using In Vitro AssayYohei Kosugi, Natalie HoseaEuropean Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|November 5, 2019
Investigation of MDR1-overexpressing cell lines to derive a quantitative prediction approach for brain disposition using in vitro efflux activitiesSho Sato, Kimio Tohyama, Yohei KosugiNeurotoxicity Research|March 17, 2025
Multi-Omics Analysis of Hippocampus in Rats Administered Trimethyltin ChlorideDouaa Zakaria, Tomoki Yamashita, Yohei KosugiJournal of Pharmaceutical Sciences|May 10, 2017
Risk Assessment Using Cytochrome P450 Time-Dependent Inhibition Assays at Single Time and Concentration in the Early Stage of Drug DiscoveryMai Kosaka, Yohei Kosugi, Hideki HirabayashiDrug Metabolism and Pharmacokinetics|November 4, 2023
Quantitation and characterization of glucosylsphingosine in cerebrospinal fluid (CSF), plasma, and brain of monkey model with Gaucher diseaseSho Sato, Shin-Ichi Matsumoto, Yohei KosugiThe AAPS Journal|June 4, 2021
Translational CNS Steady-State Drug Disposition Model in Rats, Monkeys, and Humans for Quantitative Prediction of Brain-to-Plasma and Cerebrospinal Fluid-to-Plasma Unbound Concentration RatiosSho Sato, Kota Matsumiya, Kimio Tohyama, et al.Pharmaceutical Research|August 15, 2018
Impact of P-Glycoprotein on Intestinal Absorption of an Inhibitor of Apoptosis Protein Antagonist in Rats: Mechanisms of Nonlinear Pharmacokinetics and Food EffectsSyunsuke Yamamoto, Yohei Kosugi, Hideki Hirabayashi, et al.Pageof 86