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The Journal of Experimental Medicine|June 9, 2016
Radical cure of experimental babesiosis in immunodeficient mice using a combination of an endochin-like quinolone and atovaquoneLauren A Lawres, Aprajita Garg, Vidya Kumar, et al.
Antimicrobial Agents and Chemotherapy|July 1, 2015
ELQ-300 prodrugs for enhanced delivery and single-dose cure of malariaGalen P Miley, Sovitj Pou, Rolf Winter, et al.
Journal of Medicinal Chemistry|April 12, 2014
Discovery, synthesis, and optimization of antimalarial 4(1H)-quinolone-3-diarylethersAaron Nilsen, Galen P Miley, Isaac P Forquer, et al.
ACS Infectious Diseases|June 11, 2024
3-Position Biaryl Endochin-like Quinolones with Enhanced Antimalarial PerformanceSovitj Pou, Rolf W Winter, Rozalia A Dodean, et al.
ACS Medicinal Chemistry Letters|July 16, 2025
Acridone Prodrugs with Enhanced Dual-Stage Antimalarial EfficacyRozalia A Dodean, Yuexin Li, Xiaowei Zhang, et al.
Journal of Medicinal Chemistry|June 10, 2026
Revisiting 2-Substituted-4(1<i>H</i>)-Quinolones for Targeting the <i>Plasmodium falciparum</i> Cytochrome bc<sub>1</sub> ComplexSovitj Pou, Katherine M Liebman, Rolf W Winter, et al.
Nature|May 21, 2025
In vivo screen of Plasmodium targets for mosquito-based malaria controlAlexandra S Probst, Douglas G Paton, Federico Appetecchia, et al.
Journal of Medicinal Chemistry|March 12, 2019
Discovery and Structural Optimization of Acridones as Broad-Spectrum AntimalarialsRozalia A Dodean, Papireddy Kancharla, Yuexin Li, et al.
Journal of Medicinal Chemistry|May 12, 2020
Lead Optimization of Second-Generation Acridones as Broad-Spectrum AntimalarialsPapireddy Kancharla, Rozalia A Dodean, Yuexin Li, et al.
Journal of Medicinal Chemistry|April 3, 2025
Development of Next-Generation Antimalarial Acridones with Radical Cure PotentialRozalia A Dodean, Yuexin Li, Xiaowei Zhang, et al.
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