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Medchemcomm|July 12, 2016
Covalent Tethering of Fragments For Covalent Probe DiscoveryStefan G Kathman, Alexander V StatsyukMethods in Molecular Biology (Clifton, N.J.)|May 10, 2019
Methodology for Identification of Cysteine-Reactive Covalent InhibitorsStefan G Kathman, Alexander V StatsyukJournal of Medicinal Chemistry|May 30, 2014
A fragment-based method to discover irreversible covalent inhibitors of cysteine proteasesStefan G Kathman, Ziyang Xu, Alexander V StatsyukACS Chemical Biology|March 21, 2020
Blockade of the Lysophosphatidylserine Lipase ABHD12 Potentiates Ferroptosis in Cancer CellsStefan G Kathman, Julia Boshart, Hui Jing, et al.Journal of the American Chemical Society|September 16, 2015
A Small Molecule That Switches a Ubiquitin Ligase From a Processive to a Distributive Enzymatic MechanismStefan G Kathman, Ingrid Span, Aaron T Smith, et al.Bioorganic & Medicinal Chemistry Letters|November 21, 2018
Discovery of covalent enzyme inhibitors using virtual docking of covalent fragmentsSandipan Roy Chowdhury, Steven Kennedy, Kai Zhu, et al.Chemmedchem|July 21, 2018
Structural Basis of Substrate Recognition and Covalent Inhibition of Cdu1 from Chlamydia trachomatisYesid A Ramirez, Thomas B Adler, Eva Altmann, et al.FASEB Journal : Official Publication of the Federation of American Societies for Experimental Biology|September 16, 2025
NONO Maintains SREBP-Regulated Cholesterol Biosynthesis via RNA Binding in NeuroblastomaSong Zhang, Hayley Ingram, Jack Cooper, et al.ACS Chemical Biology|March 10, 2020
Covalent-Fragment Screening of BRD4 Identifies a Ligandable Site Orthogonal to the Acetyl-Lysine Binding SitesMichael D Olp, Daniel J Sprague, Christopher J Goetz, et al.Nature Chemical Biology|March 2, 2023
Remodeling oncogenic transcriptomes by small molecules targeting NONOStefan G Kathman, Seong Joo Koo, Garrett L Lindsey, et al.Pageof 1